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14 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of Novel Indazole Derivatives as Highly Potent and Selective Humanß3-Adrenergic Receptor Agonists with the Possibility of Having No Cardiovascular Side Effects.EBI
Asahi Kasei Pharma
Discovery of 2-(1H-indazol-1-yl)-thiazole derivatives as selective EP(1) receptor antagonists for treatment of overactive bladder by core structure replacement.EBI
Asahi Kasei Pharma
Discovery of a benzimidazole series of ADAMTS-5 (aggrecanase-2) inhibitors by scaffold hopping.EBI
Asahi Kasei Pharma
SAR-based optimization of 2-(1H-pyrazol-1-yl)-thiazole derivatives as highly potent EP1 receptor antagonists.EBI
Asahi Kasei Pharma
A series of thiazole derivatives bearing thiazolidin-4-one as non-competitive ADAMTS-5 (aggrecanase-2) inhibitors.EBI
Asahi Kasei Pharma
Design of cyclic peptides with agonist activity at melanocortin receptor-4.EBI
Asahi Kasei Pharma
Discovery of selective PDE4B inhibitors.EBI
Asahi Kasei Pharma
Discovery of 4,6- and 5,7-Disubstituted Isoquinoline Derivatives as a Novel Class of Protein Kinase C ζ Inhibitors with Fragment-Merging Strategy.EBI
Asahi Kasei Pharma
The discovery of novel 3-aryl-indazole derivatives as peripherally restricted pan-Trk inhibitors for the treatment of pain.EBI
Asahi Kasei Pharma
Hit-to-lead optimization of 2-(1H-pyrazol-1-yl)-thiazole derivatives as a novel class of EP1 receptor antagonists.EBI
Asahi Kasei Pharma
Discovery of a novel 2-(1H-pyrazolo[3,4-b]pyridin-1-yl)thiazole derivative as an EPEBI
Asahi Kasei Pharma
Discovery of Novel Indazole Derivatives as Orally AvailableβEBI
Asahi Kasei Pharma
COMPOUNDS AND METHODS FOR TREATING VIRAL INFECTIONSBDB
Beth Israel Deaconess Medical Center
IMIDAZO[4,5-C]QUINOLINE COMPOUNDS AND THEIR USE AS ATM KINASE INHIBITORSBDB
Deutsches Krebsforschungszentrum