Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50001324
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276262(CHEMBL4129609)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50449137(CHEMBL3127163)
Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276250(CHEMBL4126319)
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276249(CHEMBL4126167)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276263(CHEMBL4129401)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276264(CHEMBL4128163)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276265(CHEMBL4129545)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276266(CHEMBL4126096)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276262(CHEMBL4129609)
Affinity DataKi:  8.70nMAssay Description:Antagonist activity at EP1 receptor (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276262(CHEMBL4129609)
Affinity DataKi: >2.70E+3nMAssay Description:Binding affinity to EP4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276262(CHEMBL4129609)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to EP3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50276262(CHEMBL4129609)
Affinity DataKi: >8.70E+3nMAssay Description:Binding affinity to EP2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2020
Entry Details Article
PubMed