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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 748K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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10 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery and optimization of a series of 3-(3-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amines: orally bioavailable, selective, and potent ATP-independent Akt inhibitors.EBI
Arqule
The design, preparation and SAR of novel small molecule sodium (Na(+)) channel blockers.EBI
Arqule
Potent and selective inhibitors of bacterial methionyl tRNA synthetase derived from an oxazolone-dipeptide scaffold.EBI
Arqule
The design and preparation of metabolically protected new arylpiperazine 5-HT1A ligands.EBI
Arqule
Discovery of 3-(3-(4-(1-Aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine (ARQ 092): An Orally Bioavailable, Selective, and Potent Allosteric AKT Inhibitor.EBI
Arqule
Compounds useful for inhibiting RORγtBDB
Eli Lilly
Pharmacological characterization of the nonpeptide angiotensin II receptor antagonist, U-97018.BDB
Upjohn Pharmaceuticals