65 articles for thisTarget
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Synthesis and pharmacologic evaluation of 2-endo-amino-3-exo-isopropylbicyclo[2.2.1]heptane: a potent imidazoline1 receptor specific agent.
Allergan
Synthesis and biological activity of retinoic acid receptor-alpha specific amides.
Allergan
Enantioselective syntheses of potent retinoid X receptor ligands: differential biological activities of individual antipodes.
Allergan
Phenylcyclohexene and phenylcyclohexadiene substituted compounds having retinoid antagonist activity.
Allergan
A new class of potent RAR antagonists: dihydroanthracenyl, benzochromenyl and benzothiochromenyl retinoids.
Allergan
Stereoselective synthesis and receptor activity of conformationally defined retinoid X receptor selective ligands.
Allergan
Synthesis and evaluation of 2-(arylamino)imidazoles as alpha 2-adrenergic agonists.
Allergan
Synthesis and structure-activity relationships of retinoid X receptor selective diaryl sulfide analogs of retinoic acid.
Allergan
Synthesis and evaluation of 2-[(5-methylbenz-1-ox-4-azin-6-yl)imino]imidazoline, a potent, peripherally acting alpha 2 adrenoceptor agonist.
Allergan
Synthesis and carbonic anhydrase inhibitory activity of 4-substituted 2-thiophenesulfonamides.
Allergan
Synthesis and structure-activity relationships of stilbene retinoid analogs substituted with heteroaromatic carboxylic acids.
Allergan
Synthesis and characterization of a highly potent and effective antagonist of retinoic acid receptors.
Allergan
Identification of highly potent retinoic acid receptor alpha-selective antagonists.
Allergan
Sulfuryl-substituted benzoheterocyclic derivative, preparation method and medical use thereof
Shanghai Haiyan Pharmaceutical Technology
Selective inhibitors of Alpha2-containing isoforms of Na,K-ATPase and use thereof for reduction of intraocular pressure
Yeda Research and Development
α-amino esters of hydroxypropylthiazolidine carboxamide derivative and salt form, crystal polymorph thereof
Merck Serono
Conferin, potent antioxidant and anti-inflammatory isoflavone from Caragana conferta Benth.
University of Karachi
Biochemical, cellular, and biophysical characterization of a potent inhibitor of mutant isocitrate dehydrogenase IDH1.
National Institutes of Health
Compositions and methods of inhibiting N-acylethanolamine-hydrolyzing acid amidase
University of California
Structure-based virtual screening toward the discovery of novel inhibitors of the DNA repair activity of the human apurinic/apyrimidinic endonuclease 1.
Universidade De Lisboa
Substituted pyrido[1,2-a]pyrazines for the treatment of neurodegenerative and neurological disorders
Pfizer
Biochemical and Cellular Characterization and Inhibitor Discovery of Pseudomonas aeruginosa 15-Lipoxygenase.
University of California Santa Cruz
N-((3-benzyl)-2,2-(bis-phenyl)-propan-1-amine derivatives as CETP inhibitors for the treatment of atherosclerosis and cardiovascular diseases
Bristol-Myers Squibb
Adenosine derivatives, method for the synthesis thereof, and the pharmaceutical compositions for the prevention and treatment of the inflammatory diseases containing the same as an active ingredient
Fm Therapeutics
n-Alkylboronic acid inhibitors reveal determinants of ligand specificity in the quorum-quenching and siderophore biosynthetic enzyme PvdQ.
The University of Texas
Hydroxybenzaldoximes Are D-GAP-Competitive Inhibitors of E. coli 1-Deoxy-D-Xylulose-5-Phosphate Synthase.
The Johns Hopkins University School of Medicine
Tricyclic derivative or pharmaceutically acceptable salts thereof, preparation method thereof, and pharmaceutical composition containing the same
Jeil Pharmaceutical
Dihydropyrimidin-2(1H)-one compounds as S-nitrosoglutathione reductase inhibitors
N30 Pharmaceuticals
Carboxy isatin hydrazones and their esters as Shp2 inhibitors
H. Lee Moffitt Cancer Center and Research Institute
Synthesis and investigation of dihydroxychalcones as calpain and cathepsin inhibitors.
Ewha Womans University
Bacterial thioredoxin reductase inhibitors and methods for use thereof
Thioredoxin Systems
Substituted heteroarylamine carboxamide analogs as mGluR5 negative allosteric modulators and methods of making and using the same
Vanderbilt University
Imidazopyridines and imidazopyrimidines as HIV-1 reverse transcriptase inhibitors
CSIR, Pretoria (Za)
Design and synthesis of new 2-aryl, 3-benzyl- (1,3-oxazolidine or 1,3-thiazolidine)-4-ones as selective cyclooxygenase (COX-2) inhibitor
Shahid Beheshti University
Selected C7-substituted chromone derivatives as monoamine oxidase inhibitors.
North-West University
Lipoxygenase inhibiting and antioxidant iridoids from Buddleja crispa.
Chinese Academy of Medical Sciences
The pharmacological characterization of a novel selective 5-hydroxytryptamine1A receptor antagonist, NAD-299.
Preclinical R & D, Astra Arcus
Carbonic anhydrase inhibitors: glycosylsulfanilamides act as subnanomolar inhibitors of the human secreted isoform VI.
Institut Des BiomolÉCules Max Mousseron (Ibmm)