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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine AEBI
Advinus Therapeutics
AEBI
Advinus Therapeutics
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine AEBI
Advinus Therapeutics
Rational design, synthesis, and structure-activity relationships of 5-amino-1H-pyrazole-4-carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors.EBI
Advinus Therapeutics
Discovery of pyrazole carboxylic acids as potent inhibitors of rat long chain L-2-hydroxy acid oxidase.EBI
Advinus Therapeutics
Discovery of a potent and selective small molecule hGPR91 antagonist.EBI
Advinus Therapeutics
Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors.EBI
Advinus Therapeutics
Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia.EBI
Advinus Therapeutics
Discovery and evaluation of novel FAAH inhibitors in neuropathic pain model.EBI
Advinus Therapeutics
Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions.EBI
Advinus Therapeutics
Discovery of Potent and Selective AEBI
Advinus Therapeutics
Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2's-hydroxy-3's-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors.EBI
Advinus Therapeutics
Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis.EBI
Advinus Therapeutics
Isoxazole-tethered diarylheptanoid analogs: Discovery of a new drug-like PAR2 antagonist.EBI
Advinus Therapeutics
Design and synthesis of novel xanthine derivatives as potent and selective AEBI
Advinus Therapeutics
5-alkynyl-pyrimidinesBDB
Boehringer Ingelheim International
Identification of two serine residues involved in agonist activation of the beta-adrenergic receptor.BDB
Merck Sharp and Dohme Research Laboratories
Substituted pyrrolidine-2,4-dicarboxylic acid amides as potent dipeptidyl peptidase IV inhibitors.BDB
National Health Research Institutes