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TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50067028((1E,4E)-1,5-Bis-(4-hydroxy-3-methoxy-phenyl)-penta...)
Affinity DataEC50:  900nMAssay Description:Activation of Nrf2 transcriptional activity in human LNCaP cells after 6 hrs by luciferase reporter gene assay relative to tert-butylhydroquinoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50020585(CHEMBL3290186)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of Nrf2 transcriptional activity in human LNCaP cells after 6 hrs by luciferase reporter gene assay relative to tert-butylhydroquinoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50020587(CHEMBL3290185)
Affinity DataEC50:  8.60E+3nMAssay Description:Activation of Nrf2 transcriptional activity in human LNCaP cells after 6 hrs by luciferase reporter gene assay relative to tert-butylhydroquinoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50067040(CHEMBL116438 | 1,7-bis(4-hydroxy-3-methoxyphenyl)1...)
Affinity DataEC50:  9.90E+3nMAssay Description:Activation of Nrf2 transcriptional activity in human LNCaP cells after 6 hrs by luciferase reporter gene assay relative to tert-butylhydroquinoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120402(CHEMBL3617796)
Affinity DataEC50:  1.15E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120403(CHEMBL3617798)
Affinity DataEC50:  5.00E+3nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120405(CHEMBL3617824)
Affinity DataEC50:  2.06E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120407(CHEMBL3617825)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120408(CHEMBL3617826)
Affinity DataEC50:  3.78E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120409(CHEMBL3617827)
Affinity DataEC50:  2.26E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120410(CHEMBL3617828)
Affinity DataEC50:  1.50E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120411(CHEMBL3617829)
Affinity DataEC50:  1.13E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120412(CHEMBL3617830)
Affinity DataEC50:  1.50E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120413(CHEMBL3617831)
Affinity DataEC50:  3.85E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120414(CHEMBL3617832)
Affinity DataEC50:  1.27E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120415(CHEMBL3617834)
Affinity DataEC50:  8.80E+3nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120416(CHEMBL3617835)
Affinity DataEC50:  2.45E+4nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120417(CHEMBL3617836)
Affinity DataEC50:  7.10E+3nMAssay Description:Inhibition of kelch domain of Keap1 (unknown origin) interaction to high affinity ETGE motif from Nrf2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120418(CHEMBL3617787)
Affinity DataEC50:  5.40E+3nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120419(CHEMBL3617788)
Affinity DataEC50:  1.71E+4nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120420(CHEMBL3134423)
Affinity DataEC50:  9.80E+3nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50076479(CHEMBL3235901)
Affinity DataEC50:  2.90E+3nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50109398(CHEMBL2381968)
Affinity DataEC50:  2.30E+3nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120421(CHEMBL2402206)
Affinity DataEC50:  1.18E+5nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50006931(CHEMBL2402207)
Affinity DataEC50:  2.70E+3nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50120422(CHEMBL3617852)
Affinity DataEC50:  29nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50180850(CHEMBL3819587)
Affinity DataEC50:  27nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human bronchial epithelial cells from COPD patient assessed as induction of TXNRD1 mRNA expression incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2017
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50180850(CHEMBL3819587)
Affinity DataEC50:  16nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human bronchial epithelial cells from COPD patient assessed as induction of HO-1 mRNA expression incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2017
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50180850(CHEMBL3819587)
Affinity DataEC50:  36nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human bronchial epithelial cells from COPD patient assessed as induction of GCLM mRNA expression incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2017
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50180850(CHEMBL3819587)
Affinity DataEC50:  22nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human bronchial epithelial cells from COPD patient assessed as induction of NQO1 mRNA expression incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2017
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50180850(CHEMBL3819587)
Affinity DataEC50:  12nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human BEAS2B cells assessed as induction of NQO1 specific activity incubated for 48 hrs measured on day 4 pos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2017
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212072(CHEMBL2261530)
Affinity DataEC50:  1.24E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212073(CHEMBL3952774)
Affinity DataEC50:  3.80E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212074(CHEMBL3960809)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212075(CHEMBL3970831)
Affinity DataEC50: >1.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212076(CHEMBL3962219)
Affinity DataEC50:  450nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212077(CHEMBL2261006)
Affinity DataEC50: >1.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212078(CHEMBL3926781)
Affinity DataEC50:  1.50E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212079(CHEMBL3918400)
Affinity DataEC50:  2.70E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212080(CHEMBL2261528)
Affinity DataEC50:  3.60E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataEC50:  5.40E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212081(CHEMBL3942321)
Affinity DataEC50:  1.14E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50140156(CHEMBL2387062)
Affinity DataEC50:  4.40E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212082(CHEMBL3891960)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212083(CHEMBL3943390)
Affinity DataEC50:  3.20E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM150271(US8980954, 6j)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212084(CHEMBL2261527)
Affinity DataEC50:  4.20E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212085(CHEMBL3952108)
Affinity DataEC50: >1.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212086(CHEMBL414893)
Affinity DataEC50: >1.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
University Jena

Curated by ChEMBL
LigandPNGBDBM50212087(CHEMBL3932493)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HepG2 cells after 5 hrs by ARE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2018
Entry Details Article
PubMed
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