Compile Data Set for Download or QSAR
Report error Found 6 of affinity data for UniProtKB/TrEMBL: Q9Z148
TargetHistone-lysine N-methyltransferase EHMT2(Mouse)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50202440(CHEMBL3933828)
Affinity DataKd:  1.81E+4nMAssay Description:Inhibition of His-sumo-tagged BALB/c mouse thymus histone methyltransferase G9a (969 to 1263 residues) catalytic domain expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Mouse)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50315537(chaetocin | CHEMBL1089316)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of mouse G9aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Mouse)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50315537(chaetocin | CHEMBL1089316)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of mouse Histone-lysine N-methyltransferase G9aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Mouse)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50315537(chaetocin | CHEMBL1089316)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of mouse G9aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Mouse)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50202440(CHEMBL3933828)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of His-sumo-tagged BALB/c mouse thymus histone methyltransferase G9a (969 to 1263 residues) catalytic domain expressed in Escherichia coli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Mouse)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50465081(CHEMBL4294122)
Affinity DataIC50: 7.14E+3nMAssay Description:Inhibition of mouse thymus 6His-sumo-tagged G9a (969 to 1263 residues) expressed in Escherichia coli BL21 (DE3) using histone H3 as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed