Compile Data Set for Download or QSAR
Report error Found 16 of affinity data for UniProtKB/TrEMBL: Q9Z122
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258014(N-(2-(2-(3,4-dichlorobenzylamino)-6-(4-methoxyphen...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat microsomal Delta-6-desaturaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258197(N-(2-(6-(3,4-dichlorobenzylamino)-2-(4-methoxyphen...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat microsomal Delta-6-desaturaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257757(3-(6-(3,4-dichlorobenzylamino)-2-(4-methoxyphenyl)...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat microsomal Delta-6-desaturaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257758(3-(2-(4-methoxyphenyl)-3-oxo-6-(3-(trifluoromethyl...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat microsomal Delta-6-desaturaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257808(N-(2-(6-(3,4-dichlorobenzylamino)-3-oxo-2-(pyridin...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat microsomal Delta-6-desaturaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257860(N-(2-(7-(3,4-dichlorobenzylamino)-3-(4-methoxyphen...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat microsomal Delta-6-desaturaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257919(N-(2-(7-(3,4-dichlorobenzylamino)-3-(4-methoxyphen...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat microsomal Delta-6-desaturaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257967(N-(2-(7-(4-chloro-3-(trifluoromethyl)benzylamino)-...)
Affinity DataIC50: 30nMAssay Description:Inhibition of rat microsomal Delta-6-desaturaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50535222(CHEMBL4439992)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of D6D in Sprague-Dawley rat liver microsomes using [14C]LA as substrate preincubated for 5 mins measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50116708(CHEMBL2263368)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of D6D in Sprague-Dawley rat liver microsomes using [14C]LA as substrate preincubated for 5 mins measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50298898(2-hydroxy-N-(2-(3-methyl-2-oxo-7-(3-(trifluorometh...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of stearoyl-CoA delta6 desaturase in rat microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393164(CHEMBL2153599)
Affinity DataIC50: 1.00E+8nMAssay Description:Inhibition of rat delta-6 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393165(CHEMBL2153600)
Affinity DataIC50: 1.00E+8nMAssay Description:Inhibition of rat delta-6 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393166(CHEMBL2153601)
Affinity DataIC50: 1.00E+8nMAssay Description:Inhibition of rat delta-6 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50305768(2-methyl-5-(6-(4-(2-(trifluoromethyl)phenoxy)piper...)
Affinity DataIC50: 1.00E+8nMAssay Description:Inhibition of rat delta-6 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAcyl-CoA 6-desaturase(Rat)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50362592(CHEMBL1938870)
Affinity DataIC50: 1.00E+8nMAssay Description:Inhibition of rat delta-6 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed