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Report error Found 263 of affinity data for UniProtKB/TrEMBL: Q9R1E6
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50187693(CHEMBL3186509)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant mouse ATX expressed in HEK293 cells using LPC 17:0 as substrate after 30 mins by LC-MS/MS methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50187693(CHEMBL3186509)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of recombinant mouse ATX expressed in HEK293 cells using FS3 as substrate preincubated for 15 mins followed by substrate addition measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527415(CHEMBL4529959)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM369940((R)—N-(1-(1-(1H-indazol-5-yl)-3-methyl-2,4-di...)
Affinity DataIC50: 7nMAssay Description:Inhibition of autotaxin in mouse plasma assessed as reduction in LPA (18:2) production incubated for 2 hrs LC-MS-/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527451(CHEMBL4515130)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527434(CHEMBL4466454)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527442(CHEMBL4465067)
Affinity DataIC50: 11nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM103575(ATX inhibitor 10 analogue 5 | US8551988, 65)
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50266936(CHEMBL4078601)
Affinity DataIC50: 13nMAssay Description:Inhibition of mouse ATX using TG-mTMP as substrate after 2 hrs by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2020
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527449(CHEMBL4442653)
Affinity DataIC50: 13nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527429(CHEMBL4593078)
Affinity DataIC50: 14nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527459(CHEMBL4581989)
Affinity DataIC50: 15nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527435(CHEMBL4474913)
Affinity DataIC50: 16nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527445(CHEMBL4453366)
Affinity DataIC50: 19nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50266937(CHEMBL4095125)
Affinity DataIC50: 20nMAssay Description:Inhibition of mouse ATX using TG-mTMP as substrate after 2 hrs by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2020
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527452(CHEMBL4451331)
Affinity DataIC50: 21nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM103576(ATX inhibitor 10 analogue 6)
Affinity DataIC50: 22nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50618713(CHEMBL5425421)
Affinity DataIC50: 22nMAssay Description:Inhibition of ATX in mouse plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527412(CHEMBL4482895)
Affinity DataIC50: 23nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM103577(ATX inhibitor 10 analogue 7)
Affinity DataIC50: 25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM103568(ATX inhibitor 16 | Chicago Sky Blue)
Affinity DataIC50: 26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527440(CHEMBL4469815)
Affinity DataIC50: 26nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527444(CHEMBL4438238)
Affinity DataIC50: 30nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527427(CHEMBL4572641)
Affinity DataIC50: 31nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527439(CHEMBL4471030)
Affinity DataIC50: 31nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527443(CHEMBL4534048)
Affinity DataIC50: 37nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527433(CHEMBL4515759)
Affinity DataIC50: 40nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527432(CHEMBL4474496)
Affinity DataIC50: 44nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM103980(Disubstituted aryl-Me ATX inhibitor 8)
Affinity DataIC50: 45nMAssay Description:Inhibitory activities of hit compounds towards ENPP1-5 were calculated using pNP-TMP, and the inhibitory activities of hit compounds towards ENPP6 an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50527458(CHEMBL4535941)
Affinity DataIC50: 49nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50264197(CHEMBL4094633)
Affinity DataIC50: 50nMAssay Description:Inhibition of mouse ATX-beta using LPC 16:0 as substrate by Amplex Red PLD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2020
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM103979(Disubstituted aryl-Me ATX inhibitor 7)
Affinity DataIC50: 53nMAssay Description:Inhibitory activities of hit compounds towards ENPP1-5 were calculated using pNP-TMP, and the inhibitory activities of hit compounds towards ENPP6 an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354337(2-((6-(4-(2- (azetidin-1-yl)-2- oxoethyl)piperazin...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354338(2-(4-(3-((5-cyano- 4-(4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354339((R)-2-((2-ethyl-6- (4-(2-(3- hydroxypyrrolidin- 1-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354340((S)-2-((2-ethyl-6- (4-(2-(3- hydroxypyrrolidin- 1-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354341(2-((2-ethyl-6-(4-(2- oxo-2-(pyrrolidin- 1- yl)ethy...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354342(2-(4-(3-((5-cyano- 4-(4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354343(2-((2-ethyl-6-(4-(2- morpholino-2- oxoethyl)pipera...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354344(2-((2-ethyl-6-(4-(2- (3-fluoroazetidin-1- yl)-2- o...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354345(2-((2-ethyl-6-(4-(2- (3-hydroxyazetidin- 1-yl)acet...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354353(2-((2-ethyl-6-(1-(2- (3-hydroxyazetidin- 1-yl)-2-o...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354355(2-((2-ethyl-6-(1-(2- (3-hydroxyazetidin- 1-yl)-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354356((R)-2-((2-ethyl-6- (1-(2-(3- hydroxypyrrolidin- 1-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354357((S)-2-((2-ethyl-6- (1-(2-(3- hydroxypyrrolidin- 1-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354358(2-(4-(2-ethyl-3-((4- (4- fluorophenl) thiazol-2- y...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354359(2-((2-ethyl-6-(4-(2- (3-hydroxyazetidin- 1-yl)-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354361(2-(4-(2-ethyl-3-((4- (4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354365((R)-2-(4-(2-ethyl-3- ((4-(4- fluorophenyl) thiazol...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM354366((S)-2-(4-(2-ethyl-3- ((4-(4- fluorophenyl) thiazol...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

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