Compile Data Set for Download or QSAR
Report error Found 5 of affinity data for UniProtKB/TrEMBL: Q9L4P2
TargetOXA23 carbapenemase(Acinetobacter baumannii)
Xihua University

Curated by ChEMBL
LigandPNGBDBM50339145(trans-7-oxo-6-(sulfooxy)-1,6-diazabicyclo[3.2.1]oc...)
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase OXA-23More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetOXA23 carbapenemase(Acinetobacter baumannii)
Xihua University

Curated by ChEMBL
LigandPNGBDBM50619645(NACUBACTAM | Nacubactam | FPI-1459 | RG-6080 | RG6...)
Affinity DataIC50: 4.64E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase OXA-23More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetOXA23 carbapenemase(Acinetobacter baumannii)
Xihua University

Curated by ChEMBL
LigandPNGBDBM50541448(CHEMBL4633785)
Affinity DataKi:  0.740nMAssay Description:Inhibition of Acinetobacter baumannii OXA-23 using nitrocefin as substrate preincubated for 10 mins followed by substrate addition measured every 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetOXA23 carbapenemase(Acinetobacter baumannii)
Xihua University

Curated by ChEMBL
LigandPNGBDBM50339145(trans-7-oxo-6-(sulfooxy)-1,6-diazabicyclo[3.2.1]oc...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Acinetobacter baumannii OXA-23 using nitrocefin as substrate preincubated for 10 mins followed by substrate addition measured every 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetOXA23 carbapenemase(Acinetobacter baumannii)
Xihua University

Curated by ChEMBL
LigandPNGBDBM50089084(Vaborbactam | CHEMBL3317857)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of Acinetobacter baumannii OXA-23 using nitrocefin as substrate preincubated for 10 mins followed by substrate addition measured every 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed