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Report error Found 55 of affinity data for UniProtKB/TrEMBL: Q9EQZ6
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM81292(8-Bromoadenosine 3',5'-cyclic monophosphat...)
Affinity DataEC50:  780nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50526579(CHEMBL4442766)
Affinity DataEC50:  2.36E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM81289(cid_23669773 | MLS001333136 | sodium;(4aR,6R,7R,7a...)
Affinity DataEC50:  3.87E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50526580(CHEMBL4549036)
Affinity DataEC50:  300nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50526578(CHEMBL4468490)
Affinity DataEC50:  2.06E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098793(CHEMBL3593342)
Affinity DataIC50: 900nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098793(CHEMBL3593342)
Affinity DataIC50: 900nMAssay Description:Displacement of 8-NBD-cAMP from mouse EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098792(CHEMBL3593343)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098713(CHEMBL3593335)
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241952(CHEMBL4099528)
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098719(CHEMBL3593329)
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098719(CHEMBL3593329)
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241967(CHEMBL4087626)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241953(CHEMBL4091792)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241957(CHEMBL4100650)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241961(CHEMBL4081514)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241941(CHEMBL4103080)
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241954(CHEMBL4082655)
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098712(CHEMBL3593336)
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098709(CHEMBL3593338)
Affinity DataIC50: 2.70E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098748(CHEMBL3593339)
Affinity DataIC50: 2.90E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098718(CHEMBL3593330)
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241940(CHEMBL4078805)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098797(CHEMBL3593471)
Affinity DataIC50: 3.50E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098794(CHEMBL3593341)
Affinity DataIC50: 3.60E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098710(CHEMBL3593337)
Affinity DataIC50: 4.30E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataIC50: 4.40E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241958(CHEMBL4063555)
Affinity DataIC50: 4.50E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098787(CHEMBL3593468)
Affinity DataIC50: 4.80E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098714(CHEMBL3593334)
Affinity DataIC50: 5.30E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098788(CHEMBL3593467)
Affinity DataIC50: 5.50E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098715(CHEMBL3593333)
Affinity DataIC50: 5.80E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098716(CHEMBL3593332)
Affinity DataIC50: 6.40E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098795(CHEMBL3593340)
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50241966(CHEMBL4092921)
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonist activity at mouse EPAC2 assessed as inhibition of EPAC2-mediated Rap1B (1 to 167 residues)-BODIPY GDP nucleotide exchange activity by 8-NB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2019
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098720(CHEMBL3593328)
Affinity DataIC50: 7.30E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098796(CHEMBL3593470)
Affinity DataIC50: 8.80E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataIC50: 8.90E+3nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098789(CHEMBL3593465)
Affinity DataIC50: 1.13E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098725(CHEMBL3594321)
Affinity DataIC50: 1.19E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098727(CHEMBL3594319)
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098791(CHEMBL3593344)
Affinity DataIC50: 1.90E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098798(CHEMBL3593480)
Affinity DataIC50: 2.23E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098726(CHEMBL3594320)
Affinity DataIC50: 2.24E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098721(CHEMBL3593327)
Affinity DataIC50: 2.51E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098728(CHEMBL3594318)
Affinity DataIC50: 2.65E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098786(CHEMBL3593469)
Affinity DataIC50: 2.80E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098729(CHEMBL3594317)
Affinity DataIC50: 2.83E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098724(CHEMBL3594322)
Affinity DataIC50: 3.13E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Mouse)
University Hospital Jena

Curated by ChEMBL
LigandPNGBDBM50098717(CHEMBL3593331)
Affinity DataIC50: 3.56E+4nMAssay Description:Displacement of 8-NBD-cAMP from mouse recombinant EPAC2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
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