Compile Data Set for Download or QSAR
Report error Found 4946 of affinity data for UniProtKB/TrEMBL: Q99705
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193645((E)-N-(4-amino-2-sec-butylquinolin-6-yl)-3-(4-(tri...)
Affinity DataEC50:  44nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193637((E)-N-(4-amino-2-tert-butylquinolin-6-yl)-3-(4-(tr...)
Affinity DataEC50:  29nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193613((E)-N-(4-amino-2-isopropylquinolin-6-yl)-3-(4-(tri...)
Affinity DataEC50:  160nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193617((E)-N-(4-amino-2-neopentylquinolin-6-yl)-3-(4-(tri...)
Affinity DataEC50:  110nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193620((E)-N-(4-amino-2-cyclobutylquinolin-6-yl)-3-(4-(tr...)
Affinity DataEC50:  250nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193608((E)-N-(4-(cyclobutylamino)-2-propylquinolin-6-yl)-...)
Affinity DataEC50:  270nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193611((E)-N-(4-(dimethylamino)-2-propylquinolin-6-yl)-3-...)
Affinity DataEC50:  300nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193605((E)-N-(4-amino-2-pentylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataEC50:  90nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193629((E)-N-(4-amino-2-phenylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataEC50:  6.60E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193639((E)-N-(4-methoxy-2-propylquinolin-6-yl)-3-(4-(trif...)
Affinity DataEC50:  360nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193646((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-butylph...)
Affinity DataEC50:  740nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193641((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-ethylph...)
Affinity DataEC50:  160nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193652((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-propylp...)
Affinity DataEC50:  3.60E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193626((E)-N-(4-amino-2-propylquinolin-6-yl)-3-p-tolylacr...)
Affinity DataEC50:  71nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193603((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataEC50:  61nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193627(1-(4-amino-2-propylquinolin-6-yl)-3-(4-(trifluorom...)
Affinity DataEC50:  380nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193630((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-iodophe...)
Affinity DataEC50:  280nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193635((E)-N-(4-amino-2-cyclohexylquinolin-6-yl)-3-(4-(tr...)
Affinity DataEC50:  96nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193604((E)-4-(3-(4-amino-2-propylquinolin-6-ylamino)-3-ox...)
Affinity DataEC50:  630nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193625(2-propyl-N6-(3-(4-(trifluoromethyl)phenyl)propyl)q...)
Affinity DataEC50:  1.00E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193653((E)-N-(4-amino-2-butylquinolin-6-yl)-3-(4-(trifluo...)
Affinity DataEC50:  210nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193618((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-nitroph...)
Affinity DataEC50:  310nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193621((E)-N-(2-propyl-4-(pyrrolidin-1-yl)quinolin-6-yl)-...)
Affinity DataEC50:  2.80E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193643((E)-N-(4-(azetidin-1-yl)-2-propylquinolin-6-yl)-3-...)
Affinity DataEC50:  2.50E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193606(N-(4-amino-2-propylquinolin-6-yl)-4'-chlorobipheny...)
Affinity DataEC50:  75nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193628((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(3,4-dichl...)
Affinity DataEC50:  990nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50192518(1-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)...)
Affinity DataKd:  10nMAssay Description:Antagonist activity at MCHR1 by Schild experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193609((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-fluorop...)
Affinity DataEC50:  200nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193610((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-isoprop...)
Affinity DataEC50:  520nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193615((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-chlorop...)
Affinity DataEC50:  96nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193616((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-tert-bu...)
Affinity DataEC50:  910nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193623((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(2-chlorop...)
Affinity DataEC50:  500nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193624(N-(4-amino-2-propylquinolin-6-yl)-3-(4-(trifluorom...)
Affinity DataEC50:  120nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193634(N-(4-amino-2-propylquinolin-6-yl)-4-(4-chloropheny...)
Affinity DataEC50:  370nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193636((E)-N-(4-amino-2-ethylquinolin-6-yl)-3-(4-(trifluo...)
Affinity DataEC50:  110nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50241093((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-bromoph...)
Affinity DataEC50:  93nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193640(N-(4-amino-2-propylquinolin-6-yl)-4'-(trifluoromet...)
Affinity DataEC50:  310nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50241094((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(2,4-dichl...)
Affinity DataEC50:  904nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193649(N-(4-Amino-2-methyl-quinolin-6-yl)-3-(4-trifluorom...)
Affinity DataEC50:  140nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193647((E)-N-(4-(methylamino)-2-propylquinolin-6-yl)-3-(4...)
Affinity DataEC50:  150nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193638((E)-N-(4-amino-2-cyclopentylquinolin-6-yl)-3-(4-(t...)
Affinity DataEC50:  68nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193651((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(biphenyl-...)
Affinity DataEC50:  118nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193622((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(methyl...)
Affinity DataEC50:  71nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193650((E)-N-(4-(ethylamino)-2-propylquinolin-6-yl)-3-(4-...)
Affinity DataEC50:  340nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50331161(4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-i...)
Affinity DataKd:  1.42nMAssay Description:Binding affinity to MCH-1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371872(CHEMBL257280)
Affinity DataEC50:  17nMAssay Description:Antagonist activity at MCHR1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371873(CHEMBL403730)
Affinity DataEC50:  175nMAssay Description:Antagonist activity at MCHR1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371866(CHEMBL257906)
Affinity DataEC50:  30nMAssay Description:Antagonist activity at MCHR1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371867(CHEMBL257905)
Affinity DataEC50:  69nMAssay Description:Antagonist activity at MCHR1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371868(CHEMBL269939)
Affinity DataEC50:  20nMAssay Description:Antagonist activity at MCHR1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
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