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Report error Found 21 of affinity data for UniProtKB/TrEMBL: Q99497
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597609(CHEMBL5202724)
Affinity DataIC50: 55nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597599(CHEMBL406190)
Affinity DataIC50: 63nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597613(CHEMBL5192433)
Affinity DataIC50: 85nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597598(CHEMBL5172713)
Affinity DataIC50: 118nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597603(CHEMBL5176828)
Affinity DataIC50: 118nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50589874(JYQ88)
Affinity DataIC50: 130nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PARK7 expressed in Escherichia coli BL21(DE3)Rosetta2 cells using DiFMUAc as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597611(CHEMBL5205386)
Affinity DataIC50: 180nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50589874(JYQ88)
Affinity DataIC50: 240nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PARK7 expressed in Escherichia coli BL21(DE3)Rosetta2 cells assessed as reduction in JQ-107-lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597600(CHEMBL395485)
Affinity DataIC50: 267nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597604(CHEMBL5183846)
Affinity DataIC50: 356nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597610(CHEMBL5209355)
Affinity DataIC50: 510nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597601(CHEMBL244322)
Affinity DataIC50: 676nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597612(CHEMBL5200261)
Affinity DataIC50: 700nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50448804(CHEMBL3128205)
Affinity DataIC50: 701nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597605(CHEMBL5198554)
Affinity DataIC50: 851nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597615(CHEMBL5198428)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597608(CHEMBL5200625)
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597602(CHEMBL396549)
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597606(CHEMBL5170211)
Affinity DataIC50: 2.93E+3nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597607(CHEMBL5207294)
Affinity DataIC50: 9.79E+3nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetParkinson disease protein 7(Human)
Tri-Institutional Phd Program In Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50597614(CHEMBL5184258)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of pET3a-His-tagged DJ1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in esterase activity using DiFMUAc as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed