TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.54E+4nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 890nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 620nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as induction of intracellular Ca2+ level by Fluo-4-AM dye based spectrofluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Agonist activity at rat recombinant TRPM8 receptor expressed in HEK293 cells assessed as increase in intracellular calcium concentration by fluorimet...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 7.50E+4nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as increase in current amplitude at +80 mV holding potential by whole cell patch-cla...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 4.00E+4nMAssay Description:Agonist activity at rat TRPM8 expressed in HEK293 cells assessed as increase in current amplitude at +80 mV holding potential by whole cell patch-cla...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Agonist activity at rat recombinant TRPM8 overexpressed in HEK293 cells assessed as induction of intracellular calcium influx by Fluo-4-AM dye-based ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 4.58E+4nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 4.34E+4nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 5.22E+4nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 5.10E+3nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 4.80E+3nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 850nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 440nMAssay Description:Activation of rat TRPM8 expressed in HEK293 cells assessed as stimulation of intracellular Ca2+ levelsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 2.08E+4nMAssay Description:Agonist activity at recombinant rat TRPM8 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo-4-AM probe-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.42E+4nMAssay Description:Agonist activity at recombinant rat TRPM8 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo-4-AM probe-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 1.59E+4nMAssay Description:Agonist activity at recombinant rat TRPM8 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo-4-AM probe-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataEC50: 2.61E+4nMAssay Description:Agonist activity at recombinant rat TRPM8 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo-4-AM probe-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced channel currents by whole cell patch clamp methodMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 1.80nMT: 2°CAssay Description:For functional expression of TRPM8, the full-length cDNA encoding human and rat TRPM8 are subcloned into pCI-NEO mammalian expression vectors. The ex...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced channel currents by whole cell patch clamp methodMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of intracellular calcium accumulation at 0.2 uM by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 5nMT: 2°CAssay Description:For functional expression of TRPM8, the full-length cDNA encoding human and rat TRPM8 are subcloned into pCI-NEO mammalian expression vectors. The ex...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at rat TRPM8 assessed as inhibition of menthol induced Ca2+ influx by cell-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced intracellular calcium levels preincubated for 2.5 mi...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Antagonist activity at rat TRPM8 assessed as inhibition of menthol induced Ca2+ influx by cell-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced intracellular calcium levels preincubated for 2.5 mi...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced intracellular calcium levels preincubated for 2.5 mi...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced intracellular calcium levels preincubated for 2.5 mi...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonist activity at rat TRPM8 by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced Ca2+ influx incubated 2.5 mins prior to icilin chall...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at rat TRMP8 receptor expressed in HEK293 cells assessed as menthol-induced calcium elevationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at rat TRPM8 by calcium flux assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced intracellular calcium levels preincubated for 2.5 mi...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced intracellular calcium levels preincubated for 2.5 mi...More data for this Ligand-Target Pair
