Compile Data Set for Download or QSAR
Report error Found 160 of affinity data for UniProtKB/TrEMBL: Q76JU9
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50044849(CHEMBL3311308)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity against mouse GPR40 expressed in U2OS cells by FLIPR/summary (Abse5) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50044849(CHEMBL3311308)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at mouse FFA1 receptor expressed in U2OS cells assessed as calcium mobilization after 24 hrs by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344067(rac-3-(4-(2-methyl-4-(trifluoromethyl)phenoxy)phen...)
Affinity DataEC50:  127nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344068(rac-3-(4-(2-(difluoromethoxy)-4-(trifluoromethyl)p...)
Affinity DataEC50:  77nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344069(rac-3-(4-(2-chloro-4-cyanophenoxy)phenyl)hex-4-yno...)
Affinity DataEC50:  48nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344070(rac-3-(4-(2-bromo-4-cyanophenoxy)phenyl)hex-4-ynoi...)
Affinity DataEC50:  88nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344071(rac-3-(4-(4-cyanonaphthalen-1-yloxy)phenyl)hex-4-y...)
Affinity DataEC50:  93nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344072(rac-3-(4-(4-(trifluoromethyl)naphthalen-1-yloxy)ph...)
Affinity DataEC50:  1.25E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344073(rac-3-(4-(3-chloro-5-(trifluoromethyl)pyridin-2-yl...)
Affinity DataEC50:  95nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344074(rac-3-(4-(5-bromopyrimidin-2-yloxy)phenyl)hex-4-yn...)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344075(rac-3-(4-(3-cyanopyrazin-2-yloxy)phenyl)hex-4-ynoi...)
Affinity DataEC50:  985nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344076(rac-3-(4-(isoquinolin-1-yloxy)phenyl)hex-4-ynoic a...)
Affinity DataEC50:  149nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344077(3-(4-((R)-2,3-dihydro-1H-inden-1-yloxy)phenyl)hex-...)
Affinity DataEC50:  47nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344078(rac-3-(4-(2-p-tolyl-4,5,6,7-tetrahydrobenzo[d]thia...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344079(rac-3-(4-(cyclopentyloxy)phenyl)hex-4-ynoic acid |...)
Affinity DataEC50:  124nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344080(rac-3-(4-(2-(difluoromethoxy)-4-(trifluoromethyl)p...)
Affinity DataEC50:  104nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344081(cis-rac-2-(4-(2-chloro-4-(trifluoromethyl)phenoxy)...)
Affinity DataEC50:  871nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344083(rac-5-(1-(4-(benzyloxy)phenyl)but-2-ynyl)oxazolidi...)
Affinity DataEC50:  3.71E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344084(rac-5-(1-(4-(2-(difluoromethoxy)-4-(trifluoromethy...)
Affinity DataEC50:  266nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344085(trans-rac-5-(1-(4-(2-(difluoromethoxy)-4-(trifluor...)
Affinity DataEC50:  7.06E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344086(cis-rac-5-(1-(4-(2-(difluoromethoxy)-4-(trifluorom...)
Affinity DataEC50:  136nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50344082(trans-rac-2-(4-(2-chloro-4-(trifluoromethyl)phenox...)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50343141(3-(4(2'-Methylbiphenyl-3-ylmethylamino)phenyl)prop...)
Affinity DataEC50:  19nMAssay Description:Activation of FFA1 in mouse islets assessed as glucose-dependent insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50362690(CHEMBL1829173 | AMG-837)
Affinity DataEC50:  13nMAssay Description:Agonist activity at mouse GPR40More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50207060(CHEMBL3952043)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse GPR40 assessed as increase in IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50207061(CHEMBL3980898)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse GPR40 assessed as increase in IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50434295(CHEMBL2386353)
Affinity DataEC50:  148nMAssay Description:Agonist activity at mouse FFA1 receptor transfected in human T-REX-293 cells measured for 74 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412913(CHEMBL448569)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232522(CHEMBL4065397)
Affinity DataEC50:  6.21E+3nMAssay Description:Agonist activity at mouse FFA1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267010(CHEMBL4082395)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50244066(CHEMBL4083365)
Affinity DataEC50:  54nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267051(CHEMBL4101348)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267052(CHEMBL4082459)
Affinity DataEC50:  53nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267017(CHEMBL4093180)
Affinity DataEC50: >3.30E+4nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267018(CHEMBL4065518)
Affinity DataEC50: >3.30E+4nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267019(CHEMBL4085420)
Affinity DataEC50: >3.30E+4nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267020(CHEMBL4103345)
Affinity DataEC50: >3.30E+4nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267048(CHEMBL4075190)
Affinity DataEC50: >3.30E+4nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267049(CHEMBL4095599)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267037(CHEMBL4082975)
Affinity DataEC50: >3.30E+4nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267038(CHEMBL4061093)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at GPR40 in mouse STC1 cells assessed as induction of GLP-1 secretion measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265862(CHEMBL4077507)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265865(CHEMBL4076190)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265868(CHEMBL4071228)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265875(CHEMBL4070273)
Affinity DataEC50:  8.20E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265876(CHEMBL4077353)
Affinity DataEC50:  6.10E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265898(CHEMBL4075162)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265878(CHEMBL4060517)
Affinity DataEC50:  4.50E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265899(CHEMBL4087992)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50265879(CHEMBL4065429)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
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