Compile Data Set for Download or QSAR
Report error Found 71 of affinity data for UniProtKB/TrEMBL: Q13443
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of A disintegrin and metalloprotease domain 9 (ADAM9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 56nMAssay Description:Inhibition of ADAM9 after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 56nMAssay Description:Inhibition of ADAM9 after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109614([4-(2-Ethoxy-ethoxy)-phenyl]-(3-hydroxycarbamoyl-3...)
Affinity DataIC50: 70nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109630((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 70nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50181008(TMI-05 | (S)-N-hydroxy-4-(4-(4-hydroxybut-2-ynylox...)
Affinity DataIC50: 85nMAssay Description:The molecules are dose-response tested on the following enzymes: MMP1, MMP3, MMP9, ADAM9 and ADAM10, according to the same protocol as that described...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM175095(US9115102, Apratastat)
Affinity DataIC50: 85nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50181008(TMI-05 | (S)-N-hydroxy-4-(4-(4-hydroxybut-2-ynylox...)
Affinity DataIC50: 85nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAM9 and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50453825(CHEMBL4215407 | US10556883, Compound 19a)
Affinity DataIC50: 90nMAssay Description:Inhibition of ADAM9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109631((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 180nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109610((7-Amino-3-hydroxycarbamoyl-3,4-dihydro-1H-isoquin...)
Affinity DataIC50: 190nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50370191(CHEMBL366478)
Affinity DataIC50: 230nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109635((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 260nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109629((4-Fluoro-phenyl)-(3-hydroxycarbamoyl-3,4-dihydro-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109628((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 370nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109637(4-[Ethoxy-(4-methoxy-phenyl)-phosphinoyl]-3-hydrox...)
Affinity DataIC50: 430nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50453823(CHEMBL4208519 | US10556883, Compound 19d)
Affinity DataIC50: 480nMAssay Description:Inhibition of ADAM9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109634((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 510nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109624((6-Hydroxycarbamoyl-6,7-dihydro-4H-thieno[3,2-c]py...)
Affinity DataIC50: 520nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109616((7-Hydroxycarbamoyl-7,8-dihydro-5H-pyrido[3,4-b]py...)
Affinity DataIC50: 560nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109625((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 660nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109623((4-Amino-phenyl)-(3-hydroxycarbamoyl-3,4-dihydro-1...)
Affinity DataIC50: 660nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109613((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 700nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109633((3-Hydroxycarbamoyl-1,3,4,9-tetrahydro-beta-carbol...)
Affinity DataIC50: 800nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109627((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 810nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109632((3-Fluoro-phenyl)-(3-hydroxycarbamoyl-3,4-dihydro-...)
Affinity DataIC50: 830nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109640((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 890nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109611((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 910nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109612((2-Fluoro-phenyl)-(3-hydroxycarbamoyl-3,4-dihydro-...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109615((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109622((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109639((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109621([4-(4-Amino-phenoxy)-phenyl]-(3-hydroxycarbamoyl-3...)
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109636((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109626(Biphenyl-4-yl-(3-hydroxycarbamoyl-3,4-dihydro-1H-i...)
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109620((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109638((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM379557(US9926281, Compound 36)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of ADAM-9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM113589(US8633196, 19 | US9365529, 19)
Affinity DataIC50: 3.05E+3nMAssay Description:The molecules are dose-response tested on the following enzymes: MMP1, MMP3, MMP9, ADAM9 and ADAM10, according to the same protocol as that described...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109618((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 3.11E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM175076(US9115102, Ex2)
Affinity DataIC50: 3.25E+3nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50109617((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50203527(methyl (6S,7S)-7-[(hydroxyamino)carbonyl]-6-[(4-ph...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of ADAM9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50265157((6S,7S)-N-hydroxy-5-methyl-6-(4-(5-(trifluoromethy...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of ADAM9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50575718(CHEMBL4873384)
Affinity DataIC50: 8.45E+3nMAssay Description:Inhibition of ADAM-9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM113588(US8633196, 18 | US9365529, 18)
Affinity DataIC50: 9.25E+3nMAssay Description:The molecules are dose-response tested on the following enzymes: MMP1, MMP3, MMP9, ADAM9 and ADAM10, according to the same protocol as that described...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM207973(US9266848, 11)
Affinity DataIC50: 1.00E+4nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAM9 and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2017
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM125923(US8772478, 15 | US8772478, 8)
Affinity DataIC50: 1.00E+4nMpH: 7.4Assay Description:The products are solubilized in DMSO at a concentration of 10 mM. A serial 3-fold dilution over 10 points is carried out so as to have a concentratio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM125925(US8772478, 14)
Affinity DataIC50: 1.00E+4nMpH: 7.4Assay Description:The products are solubilized in DMSO at a concentration of 10 mM. A serial 3-fold dilution over 10 points is carried out so as to have a concentratio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2014
Entry Details
Go to US Patent

TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM175083(US9115102, Ex24 | US9115102, Ex14)
Affinity DataIC50: 1.00E+4nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details
Go to US Patent

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