Compile Data Set for Download or QSAR
Report error Found 183 of affinity data for UniProtKB/TrEMBL: Q03431
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269976(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Ly...)
Affinity DataKd:  21.6nMAssay Description:Binding affinity to PTH/PTH-related peptide receptor expressed in HKRK-B28 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269976(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Ly...)
Affinity DataEC50:  26nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269971(Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  32nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269971(Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  800nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269978(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Fl...)
Affinity DataEC50:  7.20nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269977(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Ly...)
Affinity DataEC50:  20nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269976(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Ly...)
Affinity DataEC50:  2.20nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269974(Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  1.43E+3nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269973(Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  1.46E+3nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269972(Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  1.00E+3nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269978(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Fl...)
Affinity DataEC50:  0.920nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269977(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Ly...)
Affinity DataEC50:  1.10nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269976(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Ly...)
Affinity DataEC50:  0.150nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269975(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  0.0600nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269974(Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  13nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269973(Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  26nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269972(Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Ly...)
Affinity DataEC50:  53nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50318885(teriparatide | CHEMBL525610)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at PTH1R overexpressed in HEK293 cells assessed as intracellular cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50318885(teriparatide | CHEMBL525610)
Affinity DataEC50:  1nMAssay Description:Agonist activity at PTH1R overexpressed in HEK293 cells assessed as intracellular cAMP mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50318886(1,3-dibutyl-5-(diaminomethylene)pyrimidine-2,4,6(1...)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at PTH1R overexpressed in HEK293 cells assessed as intracellular cAMP mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50331020((S)-5-((2S,3S)-1-((2S,5S,8S,11S,20S)-8-((1H-imidaz...)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at recombinant PTHR1 expressed in HEK293 cells co-transfected with CRE-Luc assessed as increase of adenylyl cyclase activity after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50331021((S)-5-((2S,3S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidaz...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant PTHR1 expressed in HEK293 cells co-transfected with CRE-Luc assessed as increase of adenylyl cyclase activity after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50331022((7S,10S,13S,16S,19S,22S,25S,28S)-13-((1H-imidazol-...)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at recombinant PTHR1 expressed in HEK293 cells co-transfected with CRE-Luc assessed as increase of adenylyl cyclase activity after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246205(CHEMBL4106300)
Affinity DataEC50:  0.440nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246206(CHEMBL4090894)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246245(CHEMBL4089035)
Affinity DataEC50:  0.340nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246246(CHEMBL4067009)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246247(CHEMBL4106299)
Affinity DataEC50:  167nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246248(CHEMBL4106298)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246249(CHEMBL4063722)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246250(CHEMBL4106296)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246270(CHEMBL4088173)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246274(CHEMBL4095903)
Affinity DataEC50:  9.70nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246275(CHEMBL4073243)
Affinity DataEC50:  0.340nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246291(CHEMBL4098344)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246292(CHEMBL4078125)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246293(CHEMBL4061182)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246294(CHEMBL4071949)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246295(CHEMBL4060554)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246296(CHEMBL4098506)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246316(CHEMBL4101396)
Affinity DataEC50:  9.80nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246317(CHEMBL4063322)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246318(CHEMBL4098420)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246319(CHEMBL4080397)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246335(CHEMBL4093590)
Affinity DataEC50:  0.360nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246336(CHEMBL4106305)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246337(CHEMBL4084894)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246338(CHEMBL4063242)
Affinity DataEC50:  0.510nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246339(CHEMBL4106303)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50246362(CHEMBL4060034)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2019
Entry Details Article
PubMed
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