Compile Data Set for Download or QSAR
Report error Found 95 of affinity data for UniProtKB/TrEMBL: Q01177
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50081499(4-Hydroxy-3-[(S)-2-oxo-3-(thieno[2,3-c]pyridine-2-...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against plasmin in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50289436((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50289434((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50: 25nMAssay Description:Inhibitory concentration against plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50144535((R)-4-Oxo-1-[4-(6-phenyl-hexanoyl)-piperazine-1-ca...)
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50144551((2S,3R)-1-(4-tert-Butylcarbamoyl-piperazine-1-carb...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50076219((3S,6R)-6-Amino-6-benzyl-octahydro-indolizine-3-ca...)
Affinity DataIC50: 251nMAssay Description:Inhibitory concentration against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50144532((2S,3R)-4-Oxo-1-[4-(6-phenyl-hexanoyl)-piperazine-...)
Affinity DataIC50: 309nMAssay Description:Inhibitory activity of compound against Plasmin was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50144555((R)-1-{4-[2-(4-Benzyloxy-phenyl)-acetyl]-piperazin...)
Affinity DataIC50: 380nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50076222((1S,7S)-7-Amino-7-benzyl-hexahydro-pyrazolo[1,2-a]...)
Affinity DataIC50: 415nMAssay Description:Inhibitory concentration against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50120368((2S,3R)-1-(4-tert-Butylcarbamoyl-piperazine-1-carb...)
Affinity DataIC50: 430nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50: 873nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Lys-pNA) for plasmin in vitro.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50228840((S)-1-[(R)-2-(3,3-dimethyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibitory concentration against plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50073432(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 1.76E+3nMAssay Description:In vitro inhibitory activity was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50: 1.83E+3nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Lys-pNA) for plasmin in vitro.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50228412(methyl 1-(bis(4-acetamidophenoxy)phosphoryl)-2-(4g...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of rat plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50073429(CHEMBL84575 | CHEMBL82032 | N-((S)-1-Carbamimidoyl...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory activity was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50073431(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory activity was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50073428(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory activity was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50073427(N-((S)-1-Carbamimidoyl-2-hydroxy-piperidin-3-yl)-2...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory activity was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50073426(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory activity was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50073430(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory activity was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50289433((S)-1-((R)-2-Acetylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50073425(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory activity was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50289435((S)-1-[(R)-2-(3,3-Dimethyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against plasmin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50: 2.62E+3nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Lys-pNA) for plasmin in vitro.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50013004(CHEMBL2371636 | 2-Acetylamino-4-methyl-pentanoic a...)
Affinity DataIC50: 5.20E+3nMAssay Description:Evaluated for the inhibition of plasmin.( no inhibition at 400 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50144531(4-((2S,3R)-2-Carboxy-4-oxo-3-piperidin-4-ylmethyl-...)
Affinity DataIC50: 6.22E+3nMAssay Description:Inhibitory activity of compound against Plasmin was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50013003({1-[1-(5-Amino-1-formyl-pentylcarbamoyl)-3-methyl-...)
Affinity DataIC50: 8.90E+3nMAssay Description:Evaluated for the inhibition of plasmin.( no inhibition at 400 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140416(2-(3-Fluoro-naphthalen-2-yl)-5-methyl-2H-pyrazole-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity of compound against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140407(2-(3-Fluoro-naphthalen-2-yl)-5-methyl-2H-pyrazole-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity of compound against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50144092([4-(5-Chloro-1H-indole-2-sulfonyl)-piperazin-1-yl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against plasmin was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140367(2-(3-Methanesulfonyl-naphthalen-2-yl)-5-methyl-2H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration of compound was determined against PlasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140386(2-(6-Chloro-naphthalen-2-yl)-5-methyl-2H-pyrazole-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration of compound was determined against PlasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140380(2-(3-Fluoro-naphthalen-2-yl)-5-methyl-2H-pyrazole-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration of compound was determined against PlasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140360(2-(3-Methanesulfonyl-naphthalen-2-yl)-5-methyl-2H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration of compound was determined against PlasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140370(2-(3-Methanesulfonyl-naphthalen-2-yl)-5-methyl-2H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration of compound was determined against PlasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50142087(2'-Sulfamoyl-biphenyl-4-carboxylic acid [2-(5-brom...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against plasmin was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140424(2-(6-Chloro-naphthalen-2-yl)-5-methyl-2H-pyrazole-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity of compound against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50140413(2-(3-Fluoro-naphthalen-2-yl)-5-trifluoromethyl-2H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity of compound against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50093745((6R,7R)-7-(2-Ethoxy-benzoylamino)-7-methoxy-3-(1-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration was measured against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50228472(CHEMBL3143648)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50: 1.25E+4nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Lys-pNA) for plasmin in vitro.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50228418(methyl 1-(diphenoxyphosphoryl)-2-(4-guanidinopheny...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of rat plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50013006({1-[1-(5-Amino-1-formyl-pentylcarbamoyl)-2-phenyl-...)
Affinity DataIC50: 4.70E+4nMAssay Description:Evaluated for the inhibition of plasmin.( no inhibition at 400 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50228474(CHEMBL3143649)
Affinity DataIC50: 7.99E+4nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50013008(CHEMBL2371651 | {1-[1-(1-Formyl-4-guanidino-butylc...)
Affinity DataIC50: 8.14E+4nMAssay Description:Evaluated for the inhibition of plasmin.( no inhibition at 400 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50228473(CHEMBL3143647)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50013007(CHEMBL2371644 | {1-[1-(5-Amino-1-formyl-pentylcarb...)
Affinity DataIC50: 1.84E+5nMAssay Description:Evaluated for the inhibition of plasmin.( no inhibition at 400 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50013001({1-[1-(4-Amino-1-formyl-butylcarbamoyl)-3-methyl-b...)
Affinity DataIC50: 2.42E+5nMAssay Description:Evaluated for the inhibition of plasmin.( no inhibition at 400 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50012998(CHEMBL2371625 | {1-[1-(5-Amino-1-formyl-pentylcarb...)
Affinity DataIC50: 4.00E+5nMAssay Description:Evaluated for the inhibition of plasmin.( no inhibition at 400 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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