Compile Data Set for Download or QSAR
Report error Found 251 for UniProtKB: P51787
LigandPNGBDBM50121051(CHEMBL3621437)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human Kv7.1/KCNE1 expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50339281(5-(2,6-Dichloro-5-fluoropyridin-3-yl)-3-phenyl-2-(...)
Affinity DataEC50:  4.93E+4nMAssay Description:Activation of KCNQ1 expressed in HEK293 cells by atomic absorption Rb'+ efflux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390867(CHEMBL2070959)
Affinity DataEC50:  1.71E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390868(CHEMBL2070960)
Affinity DataEC50:  1.78E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390869(CHEMBL2070961)
Affinity DataEC50:  810nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390870(CHEMBL2070962)
Affinity DataEC50:  780nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390871(CHEMBL2070963)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390872(CHEMBL2070964)
Affinity DataEC50:  880nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390873(CHEMBL2070965)
Affinity DataEC50:  1.63E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390874(CHEMBL2070966)
Affinity DataEC50:  1.16E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390875(CHEMBL2070967)
Affinity DataEC50:  1.03E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390876(CHEMBL2070968)
Affinity DataEC50:  730nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390877(CHEMBL2070969)
Affinity DataEC50:  1.41E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390878(CHEMBL2070970)
Affinity DataEC50:  420nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390879(CHEMBL2070971)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390880(CHEMBL2070972)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390881(CHEMBL2070973)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390882(CHEMBL2070974)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390883(CHEMBL2070975)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390884(CHEMBL2070976)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390885(CHEMBL2070977)
Affinity DataEC50:  7.97E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390886(CHEMBL2070978)
Affinity DataEC50:  1.36E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390887(CHEMBL2070979)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390888(CHEMBL2070980)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390889(CHEMBL2070982)
Affinity DataEC50:  8.16E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390890(CHEMBL2070983)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390891(CHEMBL2070984)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390892(CHEMBL2070985)
Affinity DataEC50:  2.86E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390893(CHEMBL2070986)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390894(CHEMBL2070987)
Affinity DataEC50:  4.38E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390895(CHEMBL2070988)
Affinity DataEC50:  600nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390896(CHEMBL2070989)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390897(CHEMBL2070990)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390897(CHEMBL2070990)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390898(CHEMBL2070992)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390899(CHEMBL2070993)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390900(CHEMBL2070994)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390901(CHEMBL2070995)
Affinity DataEC50:  1.29E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390902(CHEMBL2070996)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390903(CHEMBL2070997)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390904(CHEMBL2070998)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390905(CHEMBL2070999)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390906(CHEMBL2071001)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390907(CHEMBL2071002)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390908(CHEMBL2071003)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390909(CHEMBL2071004)
Affinity DataEC50:  1.32E+3nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390910(CHEMBL2071005)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390911(CHEMBL2071006)
Affinity DataEC50:  2.74E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390912(CHEMBL2071007)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50390913(CHEMBL2071008)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Kv7.1 channel expressed in CHO cells assessed as depolarization-induced thallium influx after 3 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
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