Compile Data Set for Download or QSAR
Report error Found 88 of affinity data for UniProtKB/TrEMBL: P51577
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118216((4-formyl-5-hydroxy-6-methylpyridin-3-yl)methyl di...)
Affinity DataEC50:  2.19E+5nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118240(((2R,3S,4R,5R)-5-(6-amino-2-(hexylthio)-9H-purin-9...)
Affinity DataEC50:  2.00E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM, expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85043(CHEMBL69234 | CAS_149017-66-3 | NSC_6093163 | PPAD...)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM, expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336799(Suramin hexasodium | Germanin | suramin | 8,8'-[Ca...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM, expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118217(PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER | ATPga...)
Affinity DataEC50:  2.30E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  1.00E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118232(ATP, 2-meS | CHEMBL336208 | 2-MeSATP)
Affinity DataEC50:  7.40E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118226(PAPET-ATP | CHEMBL337062)
Affinity DataEC50:  1.50E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM, expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118229(MRS 2179 | CHEMBL129841)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM, expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118234(MRS 2160 | CHEMBL129904)
Affinity DataKd:  1.60E+3nMAssay Description:Dissociation constant of the compound at P2X purinoceptor 1 (P2X1) from rat vas deferens was reportedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataEC50:  2.80E+4nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118232(ATP, 2-meS | CHEMBL336208 | 2-MeSATP)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  1.00E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118221(alpha,beta-meATP | DIPHOSPHOMETHYLPHOSPHONIC ACID ...)
Affinity DataEC50:  3.30E+4nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50422739(CHEMBL413145)
Affinity DataIC50: 81nMAssay Description:Inhibitory concentration against rat P2X purinoceptor 1 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50: 233nMAssay Description:Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50: 750nMAssay Description:Antagonist activity at rat P2X4R expressed in HEK293 cells preincubated for 2 mins followed by ATP addition and measured after 4 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50: 928nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50399165(CHEMBL2180137)
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataIC50: 2.45E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataIC50: 2.45E+3nMAssay Description:Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85043(CHEMBL69234 | CAS_149017-66-3 | NSC_6093163 | PPAD...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of inward ion current elicited by ATP at rat P2X4 receptor (mutant type)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50399190(CHEMBL2180149)
Affinity DataIC50: 4.04E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50370141(TNP-ATP)
Affinity DataIC50: 4.71E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50399166(CHEMBL2180136)
Affinity DataIC50: 6.08E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118234(MRS 2160 | CHEMBL129904)
Affinity DataIC50: 9.60E+3nMAssay Description:The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) receptor from rat vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336774(sodium 1-amino-4-(3-carboxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336776(sodium 1-amino-4-(3-aminophenylamino)-9,10-dioxo-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50268685(sodium 1-amino-4-(2-carboxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50268686(sodium 1-amino-9,10-dioxo-4-(4-sulfophenylamino)-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336773(sodium 1-amino-9,10-dioxo-4-(2-sulfonatophenylamin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336772(sodium 1-amino-4-(3-bromophenylamino)-9,10-dioxo-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336771(sodium 1-amino-4-(4-fluorophenylamino)-9,10-dioxo-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336770(Sodium 1-amino-4-(4-phenoxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336769(sodium 1-amino-4-(2-ethoxyphenylamino)-9,10-dioxo-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50227023(sodium 1-amino-4-(4-methoxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336768(sodium 1-amino-4-(3-methoxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336767(PSB-716 | sodium 1-amino-4-(2-methoxyphenylamino)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50268725(sodium 1-amino-4-(4-hydroxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50268687(sodium 1-amino-4-(2-hydroxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336792(sodium 1-amino-4-(2,4-dimethylphenylamino)-9,10-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336775(sodium 1-amino-4-(4-carboxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50268635(sodium 1-amino-4-(2-aminophenylamino)-9,10-dioxo-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50268765(sodium 1-amino-4-(3-amino-5-carboxyphenylamino)-9,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50268636(Sodium 1-Amino-4-(4-aminophenylamino)-9,10-dioxo-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50227015(Sodium 1-amino-4-(4-acetylaminophenylamino)-9,10-d...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336779(sodium 1-amino-4-(3-carboxy-4-hydroxyphenylamino)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336778(Sodium 1-amino-4-[4-(diethoxyphosphoryl)methylphen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336777(sodium 1-amino-4-(4-(carboxymethyl)phenylamino)-9,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50268873(Sodium 1-amino-4-(3-amino-2,4,6-trimethylphenylami...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
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