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TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50040961(CHEMBL3354952)
Affinity DataEC50:  2.87E+4nMAssay Description:Agonist activity at mouse recombinant CB2 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429834(CHEMBL2338177)
Affinity DataEC50:  22nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429835(CHEMBL2338176)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429837(CHEMBL2338174)
Affinity DataEC50:  23nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50207795(adamantan-1-yl-(3,4-dihydro-2H-quinolin-1-yl)-meth...)
Affinity DataEC50:  126nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429836(CHEMBL2338175)
Affinity DataEC50:  28nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429838(CHEMBL2338189)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429824(CHEMBL2338188)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429825(CHEMBL2338187)
Affinity DataEC50:  51nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429826(CHEMBL2338186)
Affinity DataEC50:  19nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429827(CHEMBL2338185)
Affinity DataEC50:  50nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429828(CHEMBL2338184)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429829(CHEMBL2338183)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429830(CHEMBL2338182)
Affinity DataEC50:  7nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429831(CHEMBL2338181)
Affinity DataEC50:  40nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429845(CHEMBL2338180)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429832(CHEMBL2338179)
Affinity DataEC50:  7nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50429833(CHEMBL2338178)
Affinity DataEC50:  26nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50402865(CHEMBL2205621)
Affinity DataEC50:  50nMAssay Description:Agonist activity at mouse CB2 receptor after 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258768(CHEMBL4078901)
Affinity DataEC50:  790nMAssay Description:PAM antagonist activity at CB1 receptor in CD-1 mouse cerebellar membranes assessed as increase in [3H]CP55,940 binding after 90 mins relative to con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50303526((1-Pentyl-1H-indol-3-yl)(2,2,3,3-tetramethylcyclop...)
Affinity DataEC50:  95nMAssay Description:Inverse agonist activity at C-terminally prolink-tagged mouse CB2 receptor expressed in CHOK1 cells harboring beta-galactosidase enzyme fused beta-ar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50518025(CHEMBL4467282)
Affinity DataEC50:  15nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50518045(CHEMBL4470870)
Affinity DataEC50:  20nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50160434(AM630 | (6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-...)
Affinity DataEC50:  25nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM21282(CHEMBL306764 | 2-methyl-3-(naphthalen-1-ylcarbonyl...)
Affinity DataEC50:  160nMAssay Description:Inverse agonist activity at C-terminally prolink-tagged mouse CB2 receptor expressed in CHOK1 cells harboring beta-galactosidase enzyme fused beta-ar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50518025(CHEMBL4467282)
Affinity DataEC50:  71nMAssay Description:Inverse agonist activity at C-terminally prolink-tagged mouse CB2 receptor expressed in CHOK1 cells harboring beta-galactosidase enzyme fused beta-ar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50518046(CHEMBL4472271)
Affinity DataEC50:  1.5nMAssay Description:Inverse agonist activity at C-terminally prolink-tagged mouse CB2 receptor expressed in CHOK1 cells harboring beta-galactosidase enzyme fused beta-ar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50518046(CHEMBL4472271)
Affinity DataEC50:  52nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM21282(CHEMBL306764 | 2-methyl-3-(naphthalen-1-ylcarbonyl...)
Affinity DataEC50:  30nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50518055(CHEMBL2316263)
Affinity DataEC50:  30nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataEC50:  7.30nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataEC50:  15nMAssay Description:Inverse agonist activity at C-terminally prolink-tagged mouse CB2 receptor expressed in CHOK1 cells harboring beta-galactosidase enzyme fused beta-ar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50160434(AM630 | (6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-...)
Affinity DataEC50:  9nMAssay Description:Inverse agonist activity at C-terminally prolink-tagged mouse CB2 receptor expressed in CHOK1 cells harboring beta-galactosidase enzyme fused beta-ar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50616118(CHEMBL5421995)
Affinity DataEC50:  52nMAssay Description:Agonist activity at mouse CB2 receptor transfected in CHO-K1 cells assessed as beta2-arrestin recruitment incubated for 90 mins by luminescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50616127(CHEMBL5437134)
Affinity DataEC50:  24nMAssay Description:Agonist activity at mouse CB2 receptor transfected in CHO-K1 cells assessed as beta2-arrestin recruitment incubated for 90 mins by luminescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50616128(CHEMBL5441096)
Affinity DataEC50:  11nMAssay Description:Agonist activity at mouse CB2 receptor transfected in CHO-K1 cells assessed as beta2-arrestin recruitment incubated for 90 mins by luminescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM21244(CP-56667 [(+)-AC],XV | CP-55,940 | 2-[(1S,2S,5S)-5...)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at mouse CB2 receptor transfected in CHO-K1 cells assessed as beta2-arrestin recruitment incubated for 90 mins by luminescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50023629(CHEMBL3341861)
Affinity DataIC50: 89nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258768(CHEMBL4078901)
Affinity DataIC50: 151nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258771(CHEMBL4062376)
Affinity DataIC50: 265nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258826(CHEMBL4067016)
Affinity DataIC50: 299nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258769(CHEMBL4096928)
Affinity DataIC50: 353nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258727(CHEMBL4081259)
Affinity DataIC50: 405nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258738(CHEMBL4070648)
Affinity DataIC50: 439nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258766(CHEMBL4077975)
Affinity DataIC50: 452nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258740(CHEMBL4085844)
Affinity DataIC50: 459nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258767(CHEMBL4086756)
Affinity DataIC50: 464nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258868(CHEMBL4073727)
Affinity DataIC50: 559nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258739(CHEMBL4064299)
Affinity DataIC50: 619nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50258781(CHEMBL4099590)
Affinity DataIC50: 651nMAssay Description:Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
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