Compile Data Set for Download or QSAR
Report error Found 33 of affinity data for UniProtKB/TrEMBL: P43346
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50311609(N-((1S,3S)-3-(4-amino-5-fluoro-2-oxopyrimidin-1(2H...)
Affinity DataEC50:  90nMAssay Description:Inhibition of deoxycytidine kinase in anti CD3 and anti CD28 -stimulated mouse T cells assessed as reduction in [3H]deoxycitidine incorporationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440151(CHEMBL2426558)
Affinity DataIC50: 3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440155(CHEMBL2426598)
Affinity DataIC50: 30nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440140(CHEMBL2426588)
Affinity DataIC50: 35nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440149(CHEMBL2426560)
Affinity DataIC50: 170nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440148(CHEMBL2426561)
Affinity DataIC50: 175nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440162(CHEMBL2426591)
Affinity DataIC50: 255nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440153(CHEMBL2426460)
Affinity DataIC50: 265nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440143(CHEMBL2426585)
Affinity DataIC50: 330nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440150(CHEMBL2426559)
Affinity DataIC50: 385nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440163(CHEMBL2426590)
Affinity DataIC50: 395nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440152(CHEMBL2426557)
Affinity DataIC50: 510nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440145(CHEMBL2426583)
Affinity DataIC50: 513nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440160(CHEMBL2426593)
Affinity DataIC50: 528nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440146(CHEMBL2426582)
Affinity DataIC50: 538nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440164(CHEMBL2426589)
Affinity DataIC50: 595nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440157(CHEMBL2426596)
Affinity DataIC50: 603nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440154(CHEMBL2426459)
Affinity DataIC50: 620nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440147(CHEMBL2426581)
Affinity DataIC50: 808nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440169(CHEMBL2426578)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440159(CHEMBL2426594)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440142(CHEMBL2426586)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440161(CHEMBL2426592)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440168(CHEMBL2426577)
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440165(CHEMBL2424679)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440166(CHEMBL2426575)
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440167(CHEMBL2426576)
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440144(CHEMBL2426584)
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440156(CHEMBL2426597)
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440158(CHEMBL2426595)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440141(CHEMBL2426587)
Affinity DataIC50: 5.47E+3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440170(CHEMBL2426579)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDeoxycytidine kinase(Mouse)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50440171(CHEMBL2426580)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed