Compile Data Set for Download or QSAR
Report error Found 164 of affinity data for UniProtKB/TrEMBL: P42264
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50059674((RS)-2-amino-3-[3-hydroxy-5-(1-methyl-2H-5-tetrazo...)
Affinity DataEC50: >1.00E+6nMAssay Description:In vitro activity at Ionotropic glutamate receptor using cortical wedge assays in rat brain synaptosomaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50166286((RS)-2-amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazol...)
Affinity DataEC50:  3.50E+3nMAssay Description:In vitro activity at Ionotropic glutamate receptor using cortical wedge assays in rat brain synaptosomaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50166288((S)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5...)
Affinity DataEC50:  110nMAssay Description:In vitro activity at Ionotropic glutamate receptor using cortical wedge assays in rat brain synaptosomaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM17662(CHEMBL276815 | 2-amino-3-(3-hydroxy-5-methyl-4-iso...)
Affinity DataEC50:  3.80E+3nMAssay Description:In vitro activity at Ionotropic glutamate receptor using cortical wedge assays in rat brain synaptosomaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50166285((RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazo...)
Affinity DataEC50:  3.20E+4nMAssay Description:In vitro activity at Ionotropic glutamate receptor using cortical wedge assays in rat brain synaptosomaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50166287((RS)-2-amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetr...)
Affinity DataEC50:  7.10E+4nMAssay Description:In vitro activity at Ionotropic glutamate receptor using cortical wedge assays in rat brain synaptosomaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50059672(2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)...)
Affinity DataEC50:  330nMAssay Description:In vitro activity at Ionotropic glutamate receptor using cortical wedge assays in rat brain synaptosomaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50060627((S)-2-amino-3-(5-iodo-2,4-dioxo-3,4-dihydropyrimid...)
Affinity DataEC50:  140nMAssay Description:Potency on Ionotropic glutamate receptor kainate in dorsal root ganglion cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50069111((2S,4S)-2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioi...)
Affinity DataIC50: 380nMAssay Description:Binding affinity against Ionotropic glutamate receptor using ACPD sensitive [3H]- glutamate displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50288204((2S,3S)-3-Carboxymethyl-azetidine-2-carboxylic aci...)
Affinity DataIC50: 700nMAssay Description:Compound was tested in vitro for binding affinity against Ionotropic glutamate receptor kainate using [3H]kainate as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50069120((2S,4S)-2-Amino-4-(3,3-diphenyl-propyl)-pentanedio...)
Affinity DataIC50: 1.16E+3nMAssay Description:Binding affinity against Ionotropic glutamate receptor using ACPD sensitive [3H]- glutamate displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50069118((2S,4S)-2-Amino-4-(3-phenyl-propyl)-pentanedioic a...)
Affinity DataIC50: 1.84E+3nMAssay Description:Binding affinity against Ionotropic glutamate receptor using ACPD sensitive [3H]- glutamate displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50069118((2S,4S)-2-Amino-4-(3-phenyl-propyl)-pentanedioic a...)
Affinity DataIC50: 1.84E+3nMAssay Description:Binding affinity against Ionotropic glutamate receptor using ACPD sensitive [3H]- glutamate displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50069120((2S,4S)-2-Amino-4-(3,3-diphenyl-propyl)-pentanedio...)
Affinity DataIC50: 1.32E+4nMAssay Description:Binding affinity against Ionotropic glutamate receptor using [3H]- CGS-19755 displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50069111((2S,4S)-2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioi...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity against Ionotropic glutamate receptor using [3H]- CGS-19755 displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50017244(CHEMBL73698 | 2-Amino-3-(4-bromo-3-hydroxy-isoxazo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity of compound was determined against KA receptor, using radioligand [3H]- KAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50128264((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity of compound was determined against KA receptor, using radioligand [3H]- KAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50002370((RS)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity of compound was determined against KA receptor, using radioligand [3H]- KAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50049748(2-Amino-4-(4,4-diphenyl-butyl)-pentanedioic acid |...)
Affinity DataIC50: 1.47E+5nMAssay Description:Binding affinity against Ionotropic glutamate receptor using [3H]- CGS-19755 displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50049748(2-Amino-4-(4,4-diphenyl-butyl)-pentanedioic acid |...)
Affinity DataIC50: 1.47E+5nMAssay Description:Binding affinity against Ionotropic glutamate receptor using ACPD sensitive [3H]- glutamate displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252103(CHEMBL482097 | (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-...)
Affinity DataKi:  3.84nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50031704(2-Amino-4-methyl-pentanedioic acid | (2S,4R)-2-ami...)
Affinity DataKi:  5.69nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50207593((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxythiophe...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50002369(Digensaeure | (3S,4R)-3-(carboxymethyl)-4-(prop-1-...)
Affinity DataKi:  32.8nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426290(CHEMBL2312682)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252051((2S,4R)-2-amino-4-(3-(methylamino)-3-oxopropyl)pen...)
Affinity DataKi:  57.3nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426285(CHEMBL2312403)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426296(CHEMBL2312396)
Affinity DataKi:  185nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50126764((S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta...)
Affinity DataKi:  199nMAssay Description:Displacement of [3H]SYM from rat recombinant GluR7A expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426291(CHEMBL2312681)
Affinity DataKi:  217nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426289(CHEMBL2312683)
Affinity DataKi:  239nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50646125(CHEMBL5595349)
Affinity DataKi:  280nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426288(CHEMBL2312684)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240399(dihydrokainic acid | Dihydrokainate | (2R,3R,4S)-3...)
Affinity DataKi:  376nMAssay Description:Displacement of [3H]SYM2081 from rat cloned iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240399(dihydrokainic acid | Dihydrokainate | (2R,3R,4S)-3...)
Affinity DataKi:  376nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]SYM2081 from rat iGluR7 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  494nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  494nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252048((2S,4R)-2-amino-4-(3-methoxy-3-oxopropyl)pentanedi...)
Affinity DataKi:  1.01E+3nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50349983(CHEMBL1812596)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50295042((S)-2-Amino-3-((RS)-3-hydroxy-8-methyl-7,8-dihydro...)
Affinity DataKi:  1.38E+3nMAssay Description:Displacement of [3H]SYM from rat recombinant GluR7A expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM17660(2-amino-3-(3,5-dioxo[1,2,4]oxadiazolidin-2-yl)prop...)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50034501((S)-Amino-(3-oxo-2,3-dihydro-isoxazol-5-yl)-acetic...)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H[SYM2081 from rat recombinant GluK3a expressed in sS9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50263220(CHEMBL4075364)
Affinity DataKi:  2.15E+3nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426286(CHEMBL2312686)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50126763((S)-2-amino-3-(3-hydroxy-5-tert-butyl-4-isoxazolyl...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [3H]SYM from rat recombinant GluR7A expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50426292(CHEMBL2312402)
Affinity DataKi:  2.81E+3nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252050((2S,4R)-2-amino-4-(3-amino-3-oxopropyl)pentanedioi...)
Affinity DataKi:  2.82E+3nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252052((2S,4R)-2-amino-4-(3-(ethylamino)-3-oxopropyl)pent...)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252920((S)-1-[2'-Amino-2'-carboxyethyl]-5,7-dihydrothieno...)
Affinity DataKi:  3.25E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
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