Compile Data Set for Download or QSAR
Report error Found 4 of affinity data for UniProtKB/TrEMBL: P41738
TargetAryl hydrocarbon receptor(Rat)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50240990(NSC-721648 | 2-(3,4-dimethoxyphenyl)-5-fluorobenzo...)
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]tetrachlorodibenzo-p-dioxin from aryl hydrocarbon receptor in CRL:WI rat liver cytosolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rat)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50612693(CHEMBL5267451)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at AhR in rat liver cytosol assessed as inhibition of TCDD-induced AhR/DNA complex formation by gel retardation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Rat)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50612693(CHEMBL5267451)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of TCDD binding to rat liver cytosol AhRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Rat)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50240990(NSC-721648 | 2-(3,4-dimethoxyphenyl)-5-fluorobenzo...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]tetrachlorodibenzo-p-dioxin from aryl hydrocarbon receptor in CRL:WI rat liver cytosolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed