Compile Data Set for Download or QSAR
Report error Found 718 of affinity data for UniProtKB/TrEMBL: P30411
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093761(1-[(R)-5-Amino-1-(4-aminomethyl-benzylcarbamoyl)-p...)
Affinity DataKd:  2.80E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093760(4-Aminomethyl-N-(3-amino-propyl)-N-(2,2-dibutyl-be...)
Affinity DataKd:  1.40E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093759((R)-3-Amino-N-(4-aminomethyl-benzyl)-2-{2-[(2-cycl...)
Affinity DataKd:  1.70E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093762(3-Aminomethyl-1-(3-amino-propyl)-7-dibenzylamino-5...)
Affinity DataKd:  4.30E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093763(N-{3-[7-Dibenzylamino-3-(2-guanidino-ethyl)-2-oxo-...)
Affinity DataKd:  4.50E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093764(cyclic nonapeptide analogue | CHEMBL2369879)
Affinity DataKd:  200nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cells; 0.2-16More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093765((R)-3-Amino-N-(4-aminomethyl-benzyl)-2-{2-[(2-cycl...)
Affinity DataKd:  1.01E+5nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093767(1-(3-Aminomethyl-benzyl)-6,6-dibenzyl-1,4,5,6-tetr...)
Affinity DataKd:  7.60E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093766(((2R,4R)-2-Aminomethyl-4-benzyloxy-pyrrolidin-1-yl...)
Affinity DataKd:  6.60E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093768(5-Dibutylamino-pentanoic acid [(S)-1-(4-butyl-pyri...)
Affinity DataKd:  2.30E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093770(4-Aminomethyl-N-[(S)-1-(4-butyl-pyridin-2-yl)-2-cy...)
Affinity DataKd:  7.40E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093771(N-[(S)-1-(4-Butyl-pyridin-2-yl)-2-cyclohexyl-ethyl...)
Affinity DataKd:  5.00E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093772(N-[3-(7-Dibenzylamino-3-guanidinomethyl-2-oxo-5-ph...)
Affinity DataKd:  1.20E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093773(3-(2-Amino-ethyl)-1-(3-amino-propyl)-7-dibenzylami...)
Affinity DataKd:  1.50E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093774(N-[(2R,4R)-4-Benzyloxy-1-(naphthalene-2-carbonyl)-...)
Affinity DataKd:  1.50E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093775(5-Amino-pentanoic acid [(S)-1-(4-butyl-pyridin-2-y...)
Affinity DataKd:  6.20E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093776(4-Aminomethyl-N-(2,2-dibutyl-benzo[1,3]dioxol-4-yl...)
Affinity DataKd:  1.30E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419895(CHEMBL1956873)
Affinity DataKd:  1.58nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419897(CHEMBL1955876)
Affinity DataKd:  2.51nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419898(CHEMBL1956875)
Affinity DataKd:  2.51nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419899(CHEMBL1956876)
Affinity DataKd:  2.51nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50411275(MEN-16132 | CHEMBL218427)
Affinity DataKd:  0.0501nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419901(CHEMBL1956720)
Affinity DataKd:  0.794nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419919(CHEMBL1956721)
Affinity DataKd:  0.794nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419902(CHEMBL1956722)
Affinity DataKd:  0.316nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419904(CHEMBL1956852)
Affinity DataKd:  1.26nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419905(CHEMBL1956853)
Affinity DataKd:  0.437nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419906(CHEMBL1956854)
Affinity DataKd:  0.479nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419907(CHEMBL1956855)
Affinity DataKd:  0.724nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419908(CHEMBL1956857)
Affinity DataKd:  0.398nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419910(CHEMBL1956859)
Affinity DataKd:  0.398nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419911(CHEMBL1956860)
Affinity DataKd:  3.16nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419913(CHEMBL1956862)
Affinity DataKd:  2nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419921(CHEMBL1956864)
Affinity DataKd:  3.16nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419914(CHEMBL1956851)
Affinity DataKd:  3.16nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419915(CHEMBL1956865)
Affinity DataKd:  2.63nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419916(CHEMBL1956866)
Affinity DataKd:  1.58nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419922(CHEMBL1956870)
Affinity DataKd:  0.794nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419894(CHEMBL1956871)
Affinity DataKd:  5.01nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419923(CHEMBL1956872)
Affinity DataKd:  3.98nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419912(CHEMBL1956861)
Affinity DataKd:  1nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419903(CHEMBL1956723)
Affinity DataKd:  0.794nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419924(CHEMBL1956856)
Affinity DataKd:  0.123nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419920(CHEMBL1956863)
Affinity DataKd:  2.51nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419917(CHEMBL1956867)
Affinity DataKd:  5.01nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50419896(CHEMBL1956874)
Affinity DataKd:  3.98nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  0.0339nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataEC50:  0.0490nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50218386(CHEMBL3142416)
Affinity DataKd:  200nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cells; 0.2-16More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50293905((S)-4-amino-5-(4-(4-(2,4-dichloro-3-((2,4-dimethyl...)
Affinity DataIC50: 0.0500nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
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