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TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457473(CHEMBL4209822)
Affinity DataIC50: 30nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase using LGG as substrate after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457466(CHEMBL4206158)
Affinity DataIC50: 100nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase using LGG as substrate after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534075(CHEMBL4483393)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534075(CHEMBL4483393)
Affinity DataIC50: 3.36E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 3.43E+4nMAssay Description:Inhibition of pig kidney cytosolic Leucyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50157555(2-(3,4-dihydroxyphenyl)-4H-chromen-4-one | 3',4'-d...)
Affinity DataIC50: 3.51E+4nMAssay Description:Inhibition of pig kidney cytosolic Leucyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 4.96E+4nMAssay Description:Inhibition of pig kidney cytosolic Leucyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534077(CHEMBL4464704)
Affinity DataIC50: 6.36E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534070(CHEMBL4454667)
Affinity DataIC50: 6.83E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534074(CHEMBL4468968)
Affinity DataIC50: 6.93E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534069(CHEMBL4473220)
Affinity DataIC50: 7.68E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534072(CHEMBL4455383)
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534078(CHEMBL4557950)
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534081(CHEMBL4460083)
Affinity DataIC50: 1.63E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534071(CHEMBL4563759)
Affinity DataIC50: 3.79E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534080(CHEMBL4576374)
Affinity DataIC50: 4.09E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534073(CHEMBL4537106)
Affinity DataIC50: 7.81E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534079(CHEMBL4456116)
Affinity DataIC50: 1.11E+6nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534076(CHEMBL4435767)
Affinity DataIC50: 1.05E+6nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025043(CHEMBL3355104)
Affinity DataKi:  20nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [435-519](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50022748(2-Amino-4-methyl-pentane-1-thiol | CHEMBL69349)
Affinity DataKi:  22nMAssay Description:Competitive inhibition of LAP in porcine kidney microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025041(CHEMBL3355106)
Affinity DataKi:  39nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025042(CHEMBL3355105)
Affinity DataKi:  50nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50190111(CHEMBL327844)
Affinity DataKi:  66nMAssay Description:Inhibition of porcine LAPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  66nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  67nMAssay Description:Inhibition of porcine LAPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  67nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025070(CHEMBL3355110)
Affinity DataKi:  74nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025099(CHEMBL3355111)
Affinity DataKi:  108nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025066(CHEMBL3355109)
Affinity DataKi:  138nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025044(CHEMBL3355103)
Affinity DataKi:  157nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025050(CHEMBL3355108)
Affinity DataKi:  195nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50337147((RS)-1-amino-3-cyclohexylpropylphosphonic acid | C...)
Affinity DataKi:  210nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025047(CHEMBL3355100)
Affinity DataKi:  213nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025046(CHEMBL3355101)
Affinity DataKi:  215nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50024594(LEUCINE PHOSPHONIC ACID | (R)-1-Ammonium-3-methyl-...)
Affinity DataKi:  230nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025045(CHEMBL3355102)
Affinity DataKi:  593nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025049(CHEMBL3355107)
Affinity DataKi:  1.03E+3nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM234297(Met-ψ[P(O)(OH)CH2]-Ala (5))
Affinity DataKi:  3.64E+3nM ΔG°:  -31.0kJ/molepH: 8.4 T: 2°CAssay Description:LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50316049(1-amino-3-phenylpropylphosphonic acid | CHEMBL1090...)
Affinity DataKi:  4.55E+3nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50025048(CHEMBL3355099)
Affinity DataKi:  5.03E+3nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50170875(CHEMBL3805288)
Affinity DataKi:  7.02E+3nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50078125((1-Amino-3-phenyl-propyl)-phosphinic acid | CHEMBL...)
Affinity DataKi:  7.69E+3nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50170881(CHEMBL3805028)
Affinity DataKi:  1.52E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50170878(CHEMBL3806197)
Affinity DataKi:  1.95E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50170897(CHEMBL3805573)
Affinity DataKi:  2.08E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50170880(CHEMBL3806187)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50170884(CHEMBL3805495)
Affinity DataKi:  2.11E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
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