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Report error Found 2929 for UniProtKB: P20272
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50335938((3-benzyl-3-methyl-2,3-dihydrobenzofuran-6-yl)(pip...)
Affinity DataEC50: >1.00E+4nMAssay Description:The compound of Example 3 was tested for agonist activity at the rat CB1 (rCB1) and rCB2 receptors, at eight concentrations, in duplicate: 10, 3, 1, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM227552(US9339486, CP55,940)
Affinity DataEC50:  0.140nMAssay Description:The compound of Example 3 was tested for agonist activity at the rat CB1 (rCB1) and rCB2 receptors, at eight concentrations, in duplicate: 10, 3, 1, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  120nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061108(3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimeth...)
Affinity DataEC50:  0.0560nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061118(3-(1,1-Dimethyl-heptyl)-1-hydroxy-6,6-dimethyl-6a,...)
Affinity DataEC50:  927nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061112(9-Hydroxymethyl-6,6-dimethyl-3-pentyl-6H-benzo[c]c...)
Affinity DataEC50:  58nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061111((R)-3-(1,1-Dimethyl-heptyl)-6,6,9-trimethyl-6a,7,8...)
Affinity DataEC50:  0.580nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061113(3-(1',1'-dimethylheptyl)-6,6,9-trimethyl-6H-benzo[...)
Affinity DataEC50:  0.180nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataEC50:  11nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061110(1-Acetoxy-3-(1,1-dimethyl-heptyl)-6,6-dimethyl-6H-...)
Affinity DataEC50:  13nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061114(3-(1,1-Dimethyl-heptyl)-1-hydroxy-6,6-dimethyl-6H-...)
Affinity DataEC50:  2.40nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061109(9-Hydroxymethyl-6,6-dimethyl-3-pentyl-6a,7,10,10a-...)
Affinity DataEC50:  40nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50000727((R)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-di...)
Affinity DataEC50:  0.0350nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50010983(CHEMBL3265176)
Affinity DataEC50:  184nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50061116(3-(1,1-Dimethyl-heptyl)-1-hydroxy-9-methyl-benzo[c...)
Affinity DataEC50:  9.60nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50042912(CHEMBL3354553)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat CB1 receptor assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040960(CHEMBL3354956)
Affinity DataEC50:  5.00E+3nMAssay Description:Inverse agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50041001(CHEMBL3354942)
Affinity DataEC50:  59nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040997(CHEMBL3354946)
Affinity DataEC50:  19nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040995(CHEMBL3354948)
Affinity DataEC50:  5.40E+3nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040994(CHEMBL3354949)
Affinity DataEC50:  43nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040993(CHEMBL3354950)
Affinity DataEC50:  768nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040992(CHEMBL3354951)
Affinity DataEC50:  855nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040961(CHEMBL3354952)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040991(CHEMBL3354953)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040990(CHEMBL3354954)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040989(CHEMBL3354955)
Affinity DataEC50:  150nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040988(CHEMBL3354957)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040987(CHEMBL3354958)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040986(CHEMBL3354959)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040985(CHEMBL3354960)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040984(CHEMBL3354961)
Affinity DataEC50:  498nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040983(CHEMBL3354962)
Affinity DataEC50:  8.90E+3nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040982(CHEMBL3354963)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040981(CHEMBL3354964)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040980(CHEMBL3354965)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040979(CHEMBL3354966 | US11214548, Compound 408)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040978(CHEMBL3354967)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040977(CHEMBL3354968)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040976(CHEMBL3354969)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040975(CHEMBL3354970)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040974(CHEMBL3354971)
Affinity DataEC50:  639nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040973(CHEMBL3354972)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040972(CHEMBL3354973)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040971(CHEMBL3354974)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040970(CHEMBL3354975 | US11214548, Compound 269)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040969(CHEMBL3354976)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50040968(CHEMBL3352843)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50170333(JWH-302 | 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol...)
Affinity DataEC50:  29.3nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S binding at CB1 receptor in presence of 10 uM WIN-55212-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM50170339(JWH-251 | 1-(1-pentyl-1H-indol-3-yl)-2-o-tolyletha...)
Affinity DataEC50:  29nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S binding at CB1 receptor in presence of 10 uM WIN-55212-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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