Compile Data Set for Download or QSAR
Report error Found 619 for UniProtKB: P13631
LigandPNGBDBM31882(CHEMBL80992 | BMS184394-R)
Affinity DataKd:  75nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31884(CHEMBL81273 | BMS184394-S)
Affinity DataKd:  816nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31885(CHEMBL82089 | BMS184394)
Affinity DataKd:  64nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM31886(CHEMBL309282 | CD564)
Affinity DataKd:  3nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM31887(Ch 80 | BMS181156)
Affinity DataKd:  0.600nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM31888(CD666)
Affinity DataKd:  68nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31889(BMS 961 | BMS961 | BMS270394)
Affinity DataKd:  528nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31890(BMS270395)
Affinity DatapH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  0.200nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataKd:  0.800nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  10nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50032219(4-[(E)-2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2...)
Affinity DataEC50:  2nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article
PDB3D3D Structure (crystal)
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290184(4-(1-Isopropyl-4,4-dimethyl-1,2,3,4-tetrahydro-qui...)
Affinity DataEC50:  3nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290177(4-(4,4-Dimethyl-1,2,3,4-tetrahydro-quinolin-6-ylet...)
Affinity DataKd:  2.42E+3nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290185(4-(1-Isopropyl-4,4-dimethyl-1,2,3,4-tetrahydro-qui...)
Affinity DataKd:  72nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290180(4-(4,4-Dimethyl-1,2,3,4-tetrahydro-quinolin-7-ylet...)
Affinity DataKd:  233nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290178(4-(1-Isopropyl-4,4-dimethyl-2-oxo-1,2,3,4-tetrahyd...)
Affinity DataKd:  23nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290179(4-(1-Isopropyl-4,4-dimethyl-2-oxo-1,2,3,4-tetrahyd...)
Affinity DataKd:  17nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290182(4-(4,4-Dimethyl-2-oxo-1,2,3,4-tetrahydro-quinolin-...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290181(4-(1-Heptyl-4,4-dimethyl-1,2,3,4-tetrahydro-quinol...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290191(3-Methyl-5-[2-(5,5,8,8-tetramethyl-5,6,7,8-tetrahy...)
Affinity DataEC50:  1.15E+3nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290178(4-(1-Isopropyl-4,4-dimethyl-2-oxo-1,2,3,4-tetrahyd...)
Affinity DataEC50:  20nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290185(4-(1-Isopropyl-4,4-dimethyl-1,2,3,4-tetrahydro-qui...)
Affinity DataEC50:  6nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290179(4-(1-Isopropyl-4,4-dimethyl-2-oxo-1,2,3,4-tetrahyd...)
Affinity DataEC50:  4nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290182(4-(4,4-Dimethyl-2-oxo-1,2,3,4-tetrahydro-quinolin-...)
Affinity DataEC50:  200nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290180(4-(4,4-Dimethyl-1,2,3,4-tetrahydro-quinolin-7-ylet...)
Affinity DataEC50:  54nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  18nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290181(4-(1-Heptyl-4,4-dimethyl-1,2,3,4-tetrahydro-quinol...)
Affinity DataEC50:  260nMAssay Description:Transactivation potency for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290190((2E,4E)-3-Methyl-5-[(1R,2S)-4-methylene-2-(5,5,8,8...)
Affinity DataEC50:  355nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290192(3-Methyl-5-[5-(5,5,8,8-tetramethyl-5,6,7,8-tetrahy...)
Affinity DataEC50:  209nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290186((2E,4E)-3-Methyl-5-[(1R,2R)-1-methyl-2-(5,5,8,8-te...)
Affinity DataEC50:  1.78E+3nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50033079(4-[1-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)
Affinity DataEC50:  266nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290662((2E,4E)-3-Methyl-5-[1-(3,5,5,8,8-pentamethyl-5,6,7...)
Affinity DataEC50:  1.78E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290660((2E,4E)-3-Methyl-5-[1-(3,5,5,8,8-pentamethyl-5,6,7...)
Affinity DataEC50:  144nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50403584(CHEMBL2111534)
Affinity DataEC50: >1.00E+3nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoic acid receptor gamma using transactivatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50403583(CHEMBL2111535)
Affinity DataEC50: >1.00E+3nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoic acid receptor gamma using transactivatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  18nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoic acid receptor gamma using transactivatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075877(4-[5,5-Dimethyl-8-(5-methyl-thiophen-2-yl)-5,6-dih...)
Affinity DataKd:  11nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataEC50:  19nMAssay Description:Effective concentration for retinoic acid receptor RAR gamma transcriptional activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50120063(2,6-Difluoro-4-[(3-hydroxy-5,5,8,8-tetramethyl-5,6...)
Affinity DataEC50: >1.00E+3nMAssay Description:Effective concentration for retinoic acid receptor RAR gamma transcriptional activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  16nMAssay Description:Binding affinity for retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50097824(4-[(E)-4-(2,6,6-Trimethyl-cyclohex-1-enyl)-but-3-e...)
Affinity DataEC50:  10nMAssay Description:Ability to inhibit TTNPB-induced transactivation at retinoic acid receptor gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50097819(4-[(E)-3-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKd:  26nMAssay Description:Binding affinity towards retinoic acid receptor gamma was determined using [3H]ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50097820(4-[(E)-4-(3,3-Dimethyl-6-p-tolyl-cyclohexa-1,5-die...)
Affinity DataKd:  4nMAssay Description:Binding affinity towards retinoic acid receptor gamma was determined using [3H]ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50097821(4-{(E)-4-[2-(4-Ethyl-phenyl)-6,6-dimethyl-cyclohex...)
Affinity DataKd:  36nMAssay Description:Binding affinity towards retinoic acid receptor gamma was determined using [3H]ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  19nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  19nMAssay Description:Binding constant for baculovirus-expressed Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50029774(4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-naphthalen-2...)
Affinity DataKd:  3nMAssay Description:Binding constant for baculovirus-expressed Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  0.700nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50033079(4-[1-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)
Affinity DataKd:  887nMAssay Description:Tested for binding affinity against [3H]-ATRA binding to retinoid receptor isoform (RAR gamma) expressed in baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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