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Report error Found 12 of affinity data for UniProtKB/TrEMBL: P10599
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426066(CHEMBL2315295)
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426067(CHEMBL2315297)
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426065(CHEMBL2315294)
Affinity DataIC50: 240nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426064(CHEMBL2315292)
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426070(CHEMBL2315306)
Affinity DataIC50: 340nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426063(CHEMBL2315290)
Affinity DataIC50: 450nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426068(2-(Cyclohexyldisulfanyl)Benzo[D]Thiazole | CHEMBL2...)
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426062(CHEMBL2315288)
Affinity DataIC50: 540nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426071(CHEMBL406050 | US9018255, PX-12 | med.21724, Compo...)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50426069(CHEMBL2315305)
Affinity DataIC50: 7.31E+3nMAssay Description:Inhibition of human recombinant thioredoxin-mediated TG2 activation expressed in T84 cells assessed as blockade of 5-biotinamidopentylamine incorpora...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50407811(CHEMBL5290420)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TXN incubated for 30 mins by fluorescence based plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetThioredoxin(Human)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50366237(GAMBOGIC ACID)
Affinity DataKi:  3.11E+3nMAssay Description:Inhibition of human recombinant TRX-1 up to 60 mins by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed