Compile Data Set for Download or QSAR
Report error Found 31 of affinity data for UniProtKB/TrEMBL: P0A6I6
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82156(7-substituted pyrazoloquinolone, 15)
Affinity DataIC50: 5.00E+3nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82152(7-substituted pyrazoloquinolone, 11)
Affinity DataIC50: 5.10E+3nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82151(7-substituted pyrazoloquinolone, 10)
Affinity DataIC50: 6.20E+3nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM50517256(CHEMBL4446301)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82157(7-substituted pyrazoloquinolone, 16)
Affinity DataIC50: 7.10E+3nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82153(7-substituted pyrazoloquinolone, 12)
Affinity DataIC50: 8.80E+3nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82152(7-substituted pyrazoloquinolone, 11)
Affinity DataIC50: 1.10E+4nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82153(7-substituted pyrazoloquinolone, 12)
Affinity DataIC50: 1.30E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82156(7-substituted pyrazoloquinolone, 15)
Affinity DataIC50: 1.40E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82160(6-substituted pyrazoloquinolone, 19)
Affinity DataIC50: 1.50E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82149(7-substituted pyrazoloquinolone, 8)
Affinity DataIC50: 1.70E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82151(7-substituted pyrazoloquinolone, 10)
Affinity DataIC50: 2.20E+4nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82157(7-substituted pyrazoloquinolone, 16)
Affinity DataIC50: 4.90E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82164(6-substituted pyrazoloquinolone, 23)
Affinity DataIC50: 4.90E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82161(6-substituted pyrazoloquinolone, 20)
Affinity DataIC50: 5.40E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82155(7-substituted pyrazoloquinolone, 14)
Affinity DataIC50: 9.20E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82164(6-substituted pyrazoloquinolone, 23)
Affinity DataIC50: 9.30E+4nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM50517254(CHEMBL4553617)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM50517257(CHEMBL4584904)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82150(7-substituted pyrazoloquinolone, 9)
Affinity DataIC50: 1.03E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82165(3-substituted pyrazoloquinolone, 24)
Affinity DataIC50: 1.06E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82162(6-substituted pyrazoloquinolone, 21)
Affinity DataIC50: 1.21E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82163(6-substituted pyrazoloquinolone, 22)
Affinity DataIC50: 1.24E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82163(6-substituted pyrazoloquinolone, 22)
Affinity DataIC50: 1.25E+5nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82158(7-substituted pyrazoloquinolone, 17)
Affinity DataIC50: 1.50E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82159(4-substituted pyrazoloquinolone, 18)
Affinity DataIC50: 1.60E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82154(7-substituted pyrazoloquinolone, 13)
Affinity DataIC50: 1.66E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82161(6-substituted pyrazoloquinolone, 20)
Affinity DataIC50: 2.00E+5nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82147(7-substituted pyrazoloquinolone, 6)
Affinity DataIC50: 2.30E+5nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82148(7-substituted pyrazoloquinolone, 7)
Affinity DataIC50: 2.44E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli (strain K12))
Pfizer

LigandPNGBDBM82147(7-substituted pyrazoloquinolone, 6)
Affinity DataIC50: 2.53E+5nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2011
Entry Details Article
PubMed