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TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50052549(2-Amino-heptanedioic acid | CHEMBL111050)
Affinity DataKd:  3.00E+7nMAssay Description:Binding affinity to rat Arg IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat ARG1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat ARG1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat liver arginase using L-arginine as substrate incubated for 10 mins followed by substrate addition by scintillation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat liver arginaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of rat liver arginase using L-arginine as substrate incubated for 10 mins followed by substrate addition by scintillation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of rat ARG1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50608142(CHEMBL5281769)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of rat liver arginase using L-arginine as substrate incubated for 10 mins followed by substrate addition by scintillation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50230418(N-OMEGA-HYDROXY-L-ARGININE | Nomega-hydroxy-L-argi...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50230418(N-OMEGA-HYDROXY-L-ARGININE | Nomega-hydroxy-L-argi...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat ARG1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Sprague-Dawley rat liver arginase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50230418(N-OMEGA-HYDROXY-L-ARGININE | Nomega-hydroxy-L-argi...)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of Sprague-Dawley rat liver arginase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50608141(P-(Dihydroxyboryl)Phenylalanine | CHEMBL298071)
Affinity DataIC50: 6.00E+6nMAssay Description:Inhibition of rat liver arginase using L-arginine as substrate incubated for 10 mins followed by substrate addition by scintillation counting analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKi:  110nMAssay Description:Inhibition of N-terminal hexa-histidine tagged thrombin-cleavable rat arginase 1 expressed in Escherichia coli DE3 cells measured after 90 mins by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataKi:  500nMAssay Description:Inhibition of Sprague-Dawley rat liver arginase 1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50230418(N-OMEGA-HYDROXY-L-ARGININE | Nomega-hydroxy-L-argi...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of Sprague-Dawley rat liver arginase 1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetArginase-1(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50354832(CHEMBL1834160)
Affinity DataKi:  6.00E+4nMAssay Description:Binding affinity to rat Arg IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed