Compile Data Set for Download or QSAR
Report error Found 8 of affinity data for UniProtKB/TrEMBL: P06281
TargetRenin-1(Mouse)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM17950(CHEMBL1639 | Rasilez | (2S,4S,5S,7S)-5-amino-N-(2-...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of mouse reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetRenin-1(Mouse)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022867(2-[2-(2-{[7-(2-tert-Butoxycarbonylamino-3-phenyl-p...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin-1(Mouse)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022862(Boc-Phe-Ala-Leu-Val-Ile-His-OMe | CHEMBL101874)
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin-1(Mouse)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022864(Boc-Phe-(CH3)Ala-Leu-Val-Ile-His-OMe | CHEMBL31824...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin-1(Mouse)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022866(4-[1-{3-[1-[1-(1-amino-1-methylpropylcarboxamido)-...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin-1(Mouse)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022863(2-[2-(2-{[7-(2-tert-Butoxycarbonylamino-3-phenyl-p...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin-1(Mouse)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022865(Boc-Phe-His-Leu-Val-Ile-His-OMe | CHEMBL321937)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin-1(Mouse)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022868(2-[2-(2-{[7-(2-tert-Butoxycarbonylamino-3-phenyl-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed