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TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23564(N-(3,5-dimethylphenyl)-6-methyl-2-oxo-2H-chromene-...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23547(6,8-dichloro-2-oxo-N-phenyl-2H-chromene-3-carboxam...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23565(6,8-dichloro-N-(3-methylphenyl)-2-oxo-2H-chromene-...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23548(8-bromo-6-chloro-2-oxo-N-phenyl-2H-chromene-3-carb...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23567(8-bromo-6-chloro-N-(3-methylphenyl)-2-oxo-2H-chrom...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23536(N-cyclododecyl-6-methyl-2-oxo-2H-chromene-3-carbox...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23537(N-(adamantan-1-yl)-6-methyl-2-oxo-2H-chromene-3-ca...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23538(6-methyl-2-oxo-N-phenyl-2H-chromene-3-carboxamide ...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23539(N-benzyl-6-methyl-2-oxo-2H-chromene-3-carboxamide ...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23540(6-methyl-2-oxo-N-(2-phenylethyl)-2H-chromene-3-car...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23541(6-methyl-N-(naphthalen-1-ylmethyl)-2-oxo-2H-chrome...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23542(6-methyl-2-oxo-N-(quinolin-3-yl)-2H-chromene-3-car...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23543(2-oxo-N-phenyl-2H-chromene-3-carboxamide | JMC5219...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23545(6-nitro-2-oxo-N-phenyl-2H-chromene-3-carboxamide |...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23546(6-bromo-2-oxo-N-phenyl-2H-chromene-3-carboxamide |...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23549(6-bromo-8-methoxy-2-oxo-N-phenyl-2H-chromene-3-car...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23555(N-(2-chlorophenyl)-6-methyl-2-oxo-2H-chromene-3-ca...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23556(N-(3-chlorophenyl)-6-methyl-2-oxo-2H-chromene-3-ca...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23557(N-(4-chlorophenyl)-6-methyl-2-oxo-2H-chromene-3-ca...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23558(6-methyl-N-(2-methylphenyl)-2-oxo-2H-chromene-3-ca...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23559(6-methyl-N-(3-methylphenyl)-2-oxo-2H-chromene-3-ca...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM23560(6-methyl-N-(4-methylphenyl)-2-oxo-2H-chromene-3-ca...)
Affinity DataAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124984((R)-5-Guanidino-2-phenylmethanesulfonylamino-penta...)
Affinity DataKon:  3.10M-1s-1 Koff:  0.00000700s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50324743((3R,4R)-1-(2,2-DIFLUORO-ETHYL)-PYRROLIDINE-3,4-DIC...)
Affinity DataKd:  3.70nMAssay Description:Binding affinity to factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50324743((3R,4R)-1-(2,2-DIFLUORO-ETHYL)-PYRROLIDINE-3,4-DIC...)
Affinity DataKd:  3.70nMAssay Description:Binding affinity to factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124992(N-[(R)-4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-...)
Affinity DataKon:  0.0130M-1s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124984((R)-5-Guanidino-2-phenylmethanesulfonylamino-penta...)
Affinity DataKon:  3.10M-1s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124972(N-[4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-2-[4...)
Affinity DataKon:  0.132M-1s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124995(2-[4-(4-Chloro-benzenesulfonyl)-2-oxo-piperazin-1-...)
Affinity DataKoff:  0.00000300s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124992(N-[(R)-4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-...)
Affinity DataKoff:  0.00000200s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124990(N-[4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-2-[2...)
Affinity DataKoff:  0.00000300s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124995(2-[4-(4-Chloro-benzenesulfonyl)-2-oxo-piperazin-1-...)
Affinity DataKon:  0.190M-1s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124990(N-[4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-2-[2...)
Affinity DataKon:  0.107M-1s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124972(N-[4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-2-[4...)
Affinity DataKoff:  0.00000600s-1Assay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50537826(CHEMBL4645930)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to factor 10a (unknown origin) assessed as dissociation rate constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50537827(CHEMBL4635562)
Affinity DataKd:  1.60nMAssay Description:Binding affinity to factor 10a (unknown origin) assessed as dissociation rate constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50537828(CHEMBL4635937)
Affinity DataKd:  1.90nMAssay Description:Binding affinity to factor 10a (unknown origin) assessed as dissociation rate constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50537826(CHEMBL4645930)
Affinity DataKd:  7.5nMAssay Description:Binding affinity to factor 10a (unknown origin) by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50537827(CHEMBL4635562)
Affinity DataKd:  8.40nMAssay Description:Binding affinity to factor 10a (unknown origin) by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50537828(CHEMBL4635937)
Affinity DataKd:  10nMAssay Description:Binding affinity to factor 10a (unknown origin) by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124861(2-[2,4-bis(sulfonatooxy)phenyl]-4-oxo-3,5-bis(sulf...)
Affinity DataKd:  1.80E+3nMAssay Description:Equilibrium dissociation constant of factor Xa inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50421638(CHEMBL2303825)
Affinity DataKd:  2.00E+3nMAssay Description:Equilibrium dissociation constant of factor Xa inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124862(2-[3,4-bis(sulfonatooxy)phenyl]-4-oxo-3,5-bis(sulf...)
Affinity DataKd:  1.70E+4nMAssay Description:Equilibrium dissociation constant of factor Xa inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50421637(CHEMBL2303826)
Affinity DataKd:  9.50E+4nMAssay Description:Equilibrium dissociation constant of factor Xa inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50118798((2S,3R)-2-[3,4-bis(sulfonatooxy)phenyl]-3,5-bis(su...)
Affinity DataKd:  3.50E+3nMAssay Description:Equilibrium dissociation constant of factor Xa inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50118798((2S,3R)-2-[3,4-bis(sulfonatooxy)phenyl]-3,5-bis(su...)
Affinity DataKd:  2.61E+4nMAssay Description:Equilibrium dissociation constant of factor Xa inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50124864((2S,3S)-2-[3,4-bis(sulfonatooxy)phenyl]-3,5-bis(su...)
Affinity DataKd:  1.07E+4nMAssay Description:Equilibrium dissociation constant of factor Xa inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50266775((2R,4S)-4-(2-Chlorophenyl)-N1-(4-chlorophenyl)-4-h...)
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of human Factor-10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50266920((2R,4R)-N1-(4-Chlorophenyl)-4-ethoxy-4-ethyl-N2-(2...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of human Factor-10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Namur

LigandPNGBDBM50266921((2R,4S)-N^1^-(4-chlorophenyl)-N^2^-[2-fluoro-4-(2-...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human Factor-10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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