Compile Data Set for Download or QSAR
Report error Found 87 for UniProtKB: O09106
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50366958(CHEMBL1790587)
Affinity DataIC50: 0.400nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of mouse liver HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 2nMAssay Description:In vitro for anti-HDAC1 (Histone deacetylase 1) activity in mouse A20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50221738(CHEMBL1790595)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97708(US8476255, 96)
Affinity DataIC50: 10nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97707(US8476255, 95)
Affinity DataIC50: 10nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97695(US8476255, 55)
Affinity DataIC50: 20nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50366962(CHEMBL1790586)
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97703(US8476255, 89)
Affinity DataIC50: 30nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97698(US8476255, 59)
Affinity DataIC50: 30nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50366966(CHEMBL1790596)
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50195609(N-hydroxy-4-(3,4-dihydro-6-phenyl-4-oxopyrimidin-2...)
Affinity DataIC50: 34nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97685(US8476255, 28)
Affinity DataIC50: 36nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50002746(CHEMBL217545)
Affinity DataIC50: 36.7nMAssay Description:Inhibition of mouse HDAC1 (mean)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2014
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50234054(N-hydroxy-6-(3,4-dihydro-4-oxo-6-phenyl-2-pyrimidi...)
Affinity DataIC50: 39nMAssay Description:Inhibition of mouse liver HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50234054(N-hydroxy-6-(3,4-dihydro-4-oxo-6-phenyl-2-pyrimidi...)
Affinity DataIC50: 39nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97704(US8476255, 90)
Affinity DataIC50: 40nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97694(US8476255, 53)
Affinity DataIC50: 40nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97706(US8476255, 94)
Affinity DataIC50: 40nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50234055(N-hydroxy-5-(6-oxo-4-phenyl-1,6-dihydropyrimidin-2...)
Affinity DataIC50: 40nMAssay Description:Inhibition of mouse liver HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50234055(N-hydroxy-5-(6-oxo-4-phenyl-1,6-dihydropyrimidin-2...)
Affinity DataIC50: 40nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97697(US8476255, 58)
Affinity DataIC50: 40nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97680(US8476255, 19)
Affinity DataIC50: 42nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97700(US8476255, 77)
Affinity DataIC50: 50nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97684(US8476255, 27)
Affinity DataIC50: 50nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50002747(CHEMBL217546)
Affinity DataIC50: 50.9nMAssay Description:Inhibition of mouse HDAC1 (mean)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2014
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97688(US8476255, 32)
Affinity DataIC50: 52nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97687(US8476255, 31)
Affinity DataIC50: 54nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50195605(N-hydroxy-3-(3,4-dihydro-6-phenyl-4-oxopyrimidin-2...)
Affinity DataIC50: 57nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97686(US8476255, 29)
Affinity DataIC50: 57nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97693(US8476255, 52)
Affinity DataIC50: 60nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97701(US8476255, 84)
Affinity DataIC50: 60nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97699(BOC-LYS(AC)-AMC | US8476255, 76)
Affinity DataIC50: 60nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97683(US8476255, 24)
Affinity DataIC50: 62nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50366961(CHEMBL1790599)
Affinity DataIC50: 67nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97709(US8476255, 101)
Affinity DataIC50: 70nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM97696(US8476255, 57)
Affinity DataIC50: 70nMT: 2°CAssay Description:Assay was done in 96-well black microplate and total volume of the assay was 100 pt. Mouse liver enzyme (10 mg/ml) was diluted 1:6 with HDAC buffer. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2013
Entry Details
Go to US Patent

LigandPNGBDBM50366962(CHEMBL1790586)
Affinity DataIC50: 84nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50195615(N-hydroxy-3-(3,4-dihydro-6-benzyl-4-oxopyrimidin-2...)
Affinity DataIC50: 90nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50422364(TRAPOXIN B)
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration gainst Histone deacetylase 1 derived from NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50234114(6-(4-benzyl-6-oxo-1,6-dihydropyrimidin-2-ylthio)-N...)
Affinity DataIC50: 103nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50234114(6-(4-benzyl-6-oxo-1,6-dihydropyrimidin-2-ylthio)-N...)
Affinity DataIC50: 103nMAssay Description:Inhibition of mouse liver HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50195600(N-hydroxy-4-(3,4-dihydro-6-benzyl-4-oxopyrimidin-2...)
Affinity DataIC50: 110nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 112nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 112nMAssay Description:Inhibition of mouse liver HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 112nMAssay Description:In vitro for anti-HDAC1 (Histone deacetylase 1) activity in mouse A20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Mouse)
Institute of Technology

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 112nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Displayed 1 to 50 (of 87 total ) | Next | Last >>
Jump to: