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TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437999(CHEMBL2409452)
Affinity DataIC50: 15nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437997(CHEMBL2409457)
Affinity DataIC50: 21nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50438000(CHEMBL2409451)
Affinity DataIC50: 31nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437992(CHEMBL2409445)
Affinity DataIC50: 38nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437998(CHEMBL2409456)
Affinity DataIC50: 40nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437996(CHEMBL2409458)
Affinity DataIC50: 46nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437991(CHEMBL2409450)
Affinity DataIC50: 66nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437994(CHEMBL2409571)
Affinity DataIC50: 140nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437995(CHEMBL2409570)
Affinity DataIC50: 170nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50437993(CHEMBL2409575)
Affinity DataIC50: 370nMAssay Description:Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50111589(2-[(3,5-diiodo-4-oxidophenyl)(3,5-diiodo-4-oxocycl...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50111604(3-[1-(4-Phenoxy-phenylamino)-meth-(Z)-ylidene]-3H-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM3175(Bisindolylmaleimide 11b | Ro 31-8220 | CHEMBL6291 ...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50126829((E)-1-(6-(3-acetyl-2,4,6-trihydroxy-5-methylbenzyl...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50111585(4-bromophenylazophenol | 4-(4-Bromo-phenylazo)-phe...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50055218(1-(2-naphthlmethyl) isatin-5-carboxamide | 1-Napht...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50310357(indigo | CHEMBL599552)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50126827(4-(1-Hydroxy-naphthalen-2-ylazo)-naphthalene-1-sul...)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50023867(Indirubin)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50111591(4-[2-(2,4-Difluoro-phenylamino)-thiazol-4-yl]-benz...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50072147(CHEMBL100473 | 2,3-Bis-[1-amino-1-(2-amino-phenyls...)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM2681(3-{1-[3-(dimethylamino)propyl]-1H-indol-3-yl}-4-(1...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against Chymotrypsinogen from Thermus flavusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50284625((3R,4S)-3-Benzyl-4-bromomethyl-oxetan-2-one | CHEM...)
Affinity DataKi:  2.55E+3nMAssay Description:Inhibition of Alpha-chymotrypsin was determined by competitive substrate assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50175075((S,Z)-4-hydroxybutyl 2-cyano-3-(2-methylbenzofuran...)
Affinity DataKi:  9.42E+3nMAssay Description:Binding affinity to chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi: >1.70E+4nMAssay Description:In vitro activity against human Chymotrypsinogen B1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi: >1.70E+4nMAssay Description:Tested in vitro for inhibition of human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50152748((S)-2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carb...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50152752((S)-2-((S)-2-{(S)-3,3-Dimethyl-2-[(pyrazine-2-carb...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50152755(2-((S)-2-{(S)-3-Methoxy-2-[(pyrazine-2-carbonyl)-a...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50152753((S)-2-((S)-3,3-Dimethyl-2-{(S)-3-methyl-2-[(pyrazi...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50152754(2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carbonyl...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50152751(2-((S)-2-{(S)-2-Cyclohexyl-2-[((R)-pyrazine-2-carb...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50137733((1S,5S,6R)-2-((S)-3,3-Dimethyl-2-{(S)-3-methyl-2-[...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50152750(2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carbonyl...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50187800((S)-ethyl 1-(5-(4-phenethoxybenzyl)-1,2,4-oxadiazo...)
Affinity DataKi: >1.50E+5nMAssay Description:Binding affinity to chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50187800((S)-ethyl 1-(5-(4-phenethoxybenzyl)-1,2,4-oxadiazo...)
Affinity DataKi: >1.50E+5nMAssay Description:Inhibition of chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50410995(CHEMBL536972)
Affinity DataKi: >1.50E+5nMAssay Description:Inhibition of chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed