Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 9Q0S
TargetEpidermal growth factor receptor(Human)
University of California, Los Angeles

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50561511BDBM50561511(CHEMBL4743220)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human recombinant EGFR expressed in baculovirus infected Sf9 insect cells using poly (Glu, Tyr) 4:1 peptide as substrate incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
University of California, Los Angeles

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50561511BDBM50561511(CHEMBL4743220)
Affinity DataIC50: 4nMAssay Description:Inhibition of wild type EGFR in human U87 cells assessed as heparin/human EGF stimulated phosphorylation after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)