Affinity DataKi: 79nMAssay Description:Inhibition of [3H]norepinephrine uptake at the rat norepinephrine transporter.More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 79nMAssay Description:Compound was tested for the inhibition of norepinephrine (NE) reuptakeMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Inhibition of [3H]NE uptake in NET in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Inhibition of rat brain Norepinephrine transporter as accumulation of [3H]-NEMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of [3H]-5-norepinephrine reuptake in human NET expressed in HEK293 cells by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of re-uptake of [3H]-NE at human NET expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Inhibition of rat brain Norepinephrine transporter as accumulation of [3H]NEMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:NET: This protocol was designed to measure inhibition of uptake by the human norepinephrine transporter. The reagents were human NET (HEK293F) cells,...More data for this Ligand-Target Pair
Affinity DataIC50: 496nMAssay Description:Inhibition of binding of [3H]nisoxetine to (NET) norepinephrine transporter in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 496nMAssay Description:Binding affinity at the norepinephrine transporter in rat striatum by [3H]nisoxetine displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 496nMAssay Description:Inhibition of binding of [3H]- nisoxatine to Norepinephrine transporter (NET) of rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 496nMAssay Description:Displacement of [3H]nisoxetine from NET in Sprague-Dawley rat brain cortex membranes after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 496nMAssay Description:Affinity at norepinephrine transporter (NET) in rat striatum, using [3H]- nisoxatine as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 496nMAssay Description:Inhibition of [3H]nisoxetine binding to norepinephrine transporter of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 496nMAssay Description:Binding affinity towards norepinephrine transporter in rat striatum using [3H]nisoxetine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.27E+3nMAssay Description:The compound was tested for binding affinity nisoxatine ligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.27E+3nMAssay Description:Displacement of [3H]nisoxetine from rat brain norepinephrine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 1.27E+3nMAssay Description:Binding affinity at norepinephrine transporter using [3H]nisoxetine as radioligand from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of human NET expressed in HEK293 cells assessed as inhibition of noradrenaline reuptake after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:In vitro binding affinity towards Norepinephrine transporter rat cerebral cortical homogenates by [3H]nisoxetine displacement.More data for this Ligand-Target Pair
