Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 9FJX
TargetProtein cereblon(Human)
Max Planck Institute For Developmental Biology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026472BDBM50026472((methanesulfinyl)methanedimethyl sulfoxide | CHEMB...)
Affinity DataKi:  1.37E+5nMAssay Description:Binding affinity to human CRBN-thalidomide binding domain expressed in Escherichia coli by measuring baseline corrected normalized fluorescence by MS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein cereblon(Human)
Max Planck Institute For Developmental Biology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026472BDBM50026472((methanesulfinyl)methanedimethyl sulfoxide | CHEMB...)
Affinity DataIC50: 2.64E+5nMAssay Description:Binding affinity to human CRBN-thalidomide binding domain expressed in Escherichia coli by measuring baseline corrected normalized fluorescence by MS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein cereblon(Human)
Max Planck Institute For Developmental Biology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026472BDBM50026472((methanesulfinyl)methanedimethyl sulfoxide | CHEMB...)
Affinity DataKi:  1.37E+8nMAssay Description:Competitive binding affinity to human CRBN-thalidomide binding domain expressed in Escherichia coli by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)