| Details for Substrate
Dual specificity mitogen-activated protein kinase kinase 1 [K97R] without Explicit Binding Affinity Data |
| Binding Enzyme 1: | RAF proto-oncogene serine/threonine-protein kinase [Y340E,Y341E] |
| Binding Enzyme 2: | RAF proto-oncogene serine/threonine-protein kinase [1-324] |
| Binding Enzyme 3: | Serine/threonine-protein kinase B-raf [V600E] |
| Binding Enzyme 4: | RAF proto-oncogene serine/threonine-protein kinase |
| Synonyms: |
MEK1 (K97R)
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Dual specificity mitogen-activated protein kinase kinase 1 (MEK1)(K97R)
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MP2K1_HUMAN
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MAP2K1
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MEK1
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PRKMK1
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| Type: | n/a |
| Topology: | n/a |
| Mol. Mass.: | 43467.04 Dalton |
| Organism: | Human |
| Description: | Biotinylated full length MEK1 with an inactivating K97R ATP binding site mutation. |
| Residue: | 393 |
| Sequence: | MPKKKPTPIQLNPAPDGSAVNGTSSAETNLEALQKKLEELELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARRLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFGCQVEGDAAETPPRPRTPGRPLSSYGMDSRPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLNQPSTPTHAAGV |
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