Assay Method Information

Assay Name:  ChEMBL_2250136 (CHEMBL5164346)
Description:  Antagonist activity at human MC4R transfected in HEK293 cells co-transfected with GScAMP22F assessed as decrease in alpha-MSH induced cAMP level in presence of 70 nM alpha-MSH by split luciferase cAMP sensor dynamic assay
Affinity data for this assay
 

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