| Assay Method Information | |
| | ChEMBL_946850 (CHEMBL2345515) |
| Description: | Competitive inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as inhibition constant for dissociation of enzyme-inhibitor complex incubated for 15 mins prior to substrate addition measured after 45 mins by fluorescence assay |
| Affinity data for this assay | |
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