Assay Method Information

Assay Name:  ChEMBL_1809732 (CHEMBL4309192)
Description:  Antagonist activity at prolink-tagged TrkB (unknown origin) expressed in cells assessed as inhibition of BDNF-induced receptor phosphorylation by measuring reduction in EA-tagged SH2 protein recruitment preincubated for 30 mins followed by BDNF addition measured after 2 hrs by PathHunter enzyme complementation assay
Affinity data for this assay
 

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