| Assay Method Information | |
| | ChEMBL_1870580 (CHEMBL4371747) |
| Description: | Competitive inhibition of human GAT1 expressed in COS cells assessed as reduction in [2H6]GABA uptake by measuring [2H6]GABA Kd(app) at 1 uM preincubated for 25 mins followed by [2H6]GABA addition and measured after 4 mins by liquid scintillation counting method (Rvb = 28.3 +/- 1.5 nM) |
| Affinity data for this assay | |
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