Assay Method Information

Assay Name:  ChEMBL_1718153 (CHEMBL4133153)
Description:  Antagonist activity at P2X7 receptor in Swiss mouse peritoneal macrophages assessed as inhibition of BzATP-induced current at holding potential of -60 mV preincubated for 5 mins followed by BzATP addition measured after 5 mins by Whole cell patch-clamp analysis
Affinity data for this assay
 

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