Assay Method Information | |
| ChEMBL_1654447 (CHEMBL4003813) |
Description: | Antagonist activity at human adenosine A1 receptor expressed in HEK293 cell membranes assessed as decrease in CPA/forskolin-induced cAMP level pretreated for 15 mins followed by agonist addition for 15 mins and subsequent forskolin stimulation measured after 30 mins |
Affinity data for this assay | |
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