Assay Method Information

Assay Name:  ChEMBL_985752 (CHEMBL2433969)
Description:  Antagonist activity at rat recombinant TRPM8 overexpressed in HEK293 cells assessed as inhibition of icilin-induced intracellular calcium influx preincubated for 5 mins followed by icilin challenge by Fluo-4-AM dye-based spectrofluorimetric analysis
Affinity data for this assay
 

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