| Assay Method Information | |
| | ChEMBL_2194228 (CHEMBL5106588) |
| Description: | Antagonist activity at D4R (unknown origin) expressed in human HEK293T cells assessed as inhibition of dopamine-induced Gi protein activation pretreated for 10 mins followed by dopamine addition and measured after 2.5 mins by BRET assay |
| Affinity data for this assay | |
|---|---|
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