Assay Method Information

Assay Name:  ChEMBL_2194227 (CHEMBL5106587)
Description:  Antagonist activity at D4R (unknown origin) expressed in human HEK293T cells assessed as inhibition of dopamine-induced G0 protein activation pretreated for 10 mins followed by dopamine addition and measured after 2.5 mins by BRET assay
Affinity data for this assay
 

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