| Assay Method Information | |
| | ChEMBL_1541711 (CHEMBL3745219) |
| Description: | Antagonist activity at P2X7 receptor in human lymphocytes assessed as inhibition of ATP-induced ethidium ion uptake preincubated for 5 mins followed by ATP addition and incubated further 2 mins prior to ethidium addition measured up to 5 mins by flow cytometric analysis |
| Affinity data for this assay | |
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