| Assay Method Information | |
| | Inhibitory Effect on the Enzymatic Activity of KLK |
| Description: | Table 4: The molecules were tested in order to evaluate their possible inhibitory effect on the enzymatic activity of KLK1. The % inhibitions were determined from the residual activity of the hydrolysis of the Boc-PFR-AMC fluorogenic substrate (100 μM) by KLK1 (1.6 nM) after 15 minutes of incubation at 37° C. with each molecule at 10 μM. |
| Affinity data for this assay | |
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